SCHEMBL1901540

SCHEMBL1901540

c1ccc(CCCCNc2ncnc3sccc23)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 6/20 0.62
SMN1; SMN2 Q16637 4/20 0.62
LMNA P02545 5/20 0.57
NPC1 O15118 2/20 0.55
TSHR P16473 2/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
RAB9A P51151 3/20 0.53
GALR3 O60755 1/20 0.53
NR2F2 P24468 1/20 0.53
PIK3CD O00329 1/20 0.51
PIK3R1 P27986 1/20 0.51
TNF P01375 2/20 0.50
NOD1 Q9Y239 2/20 0.50
HSD17B10 Q99714 1/20 0.50
EGFR P00533 1/20 0.50
APP P05067 1/20 0.50
MAPK1 P28482 1/20 0.50
ALDH1A1 P00352 1/20 0.48
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8506192 0.96 HTT (0.63) HTTSMN1; SMN2LMNANPC1TSHR
SCHEMBL1904097 0.91 HTT (0.70) HTTSMN1; SMN2LMNANPC1TSHR
SCHEMBL11500313 0.81 SMN1; SMN2 (0.56) HTTSMN1; SMN2LMNANPC1TSHR
SCHEMBL9607949 0.79 HTT (0.55) HTTSMN1; SMN2LMNANPC1TSHR
SCHEMBL13948948 0.78 LMNA (0.81) HTTSMN1; SMN2LMNATSHRMEN1
SCHEMBL8505732 0.77 HTT (0.63) HTTSMN1; SMN2LMNANPC1TSHR
SCHEMBL10914077 0.77 RAB9A (0.63) HTTSMN1; SMN2LMNANPC1TSHR
SCHEMBL3966396 0.77 HTT (0.68) HTTSMN1; SMN2LMNANPC1TSHR
SCHEMBL8505626 0.77 HTT (0.68) HTTSMN1; SMN2LMNANPC1TSHR
SCHEMBL8516166 0.77 HTT (0.77) HTTSMN1; SMN2LMNANPC1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2320904-A2 AMINOPYRIMIDINE INHIBITORS OF HISTAMINE RECEPTORS FOR THE TREATMENT OF DISEASE Kalypsys, Inc. (US) 2011-05-18 EP disclosed
WO-2010030757-A2 AMINOPYRIMIDINE INHIBITORS OF HISTAMINE RECEPTORS FOR THE TREATMENT OF DISEASE KALYPSYS INC. (US) 2010-03-18 WO disclosed