SCHEMBL19036787

SCHEMBL19036787

Cn1c(=O)c2c(ncn2COCN)n(C)c1=O

nearest known ligand 0.69

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 11/20 0.69
LMNA P02545 4/20 0.61
MAPT P10636 1/20 0.61
SMN1; SMN2 Q16637 4/20 0.58
RXFP1 Q9HBX9 1/20 0.56
MAPK1 P28482 1/20 0.54
POLB P06746 1/20 0.54
ALDH1A1 P00352 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11374923 0.87 ADORA2B (0.62) ADORA2BLMNAMAPTSMN1; SMN2RXFP1
SCHEMBL19036507 0.85 ADORA2B (0.68) ADORA2BLMNAMAPTSMN1; SMN2RXFP1
SCHEMBL11380544 0.84 ADORA2B (0.59) ADORA2BLMNAMAPTSMN1; SMN2RXFP1
SCHEMBL13659055 0.84 SMN1; SMN2 (0.66) ADORA2BLMNAMAPTSMN1; SMN2RXFP1
Dimethylamine SCHEMBL11381767 0.83 SMN1; SMN2 (0.59) ADORA2BLMNAMAPTSMN1; SMN2RXFP1
SCHEMBL8666393 0.83 ADORA2B (0.79) ADORA2BLMNAMAPTSMN1; SMN2RXFP1
SCHEMBL11377411 0.82 ADORA2B (0.59) ADORA2BLMNAMAPTRXFP1
SCHEMBL4516866 0.82 ADORA2B (1.00) ADORA2BLMNAMAPTSMN1; SMN2RXFP1
SCHEMBL16120984 0.81 ADORA2B (0.81) ADORA2BLMNAMAPTSMN1; SMN2RXFP1
SCHEMBL11383083 0.81 SMN1; SMN2 (0.63) ADORA2BLMNAMAPTSMN1; SMN2RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3184527-A1 2,6-DIOXO,-2,3-DIHYDRO-1H-PURINE COMPOUNDS USEFUL FOR TREATING DISORDERS RELATED TO THE ACTIVITY OF THE TRPA1 CHANNEL Hydra Biosciences, Inc. (US) 2017-06-28 EP disclosed