SCHEMBL19045790

SCHEMBL19045790

COC(=O)c1cnn2cc(C)cnc12

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 13/20 0.57
HSD11B1 P28845 3/20 0.51
PDE10A Q9Y233 3/20 0.49
PDE3A Q14432 1/20 0.49
ALDH1A1 P00352 3/20 0.46
LMNA P02545 2/20 0.46
KDM4E B2RXH2 2/20 0.46
HSD17B10 Q99714 2/20 0.46
HPGD P15428 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17781274 0.85 KDM4E (0.57) PDE2APDE10APDE3AALDH1A1KDM4E
SCHEMBL310126 0.83 PDE2A (0.59) PDE2AHSD11B1PDE10APDE3AALDH1A1
SCHEMBL19029939 0.83 LMNA (0.47) PDE2AHSD11B1ALDH1A1LMNAKDM4E
SCHEMBL10071025 0.83 LMNA (0.44) PDE2APDE10APDE3AALDH1A1LMNA
SCHEMBL21326698 0.81 PDE2A (0.53) PDE2AHSD11B1PDE10APDE3A
SCHEMBL19029896 0.81 PDE2A (0.45) PDE2APDE10APDE3AALDH1A1LMNA
SCHEMBL30579399 0.75 LMNA (0.45) PDE2AALDH1A1LMNAKDM4EHSD17B10
SCHEMBL19030768 0.75 LMNA (0.72) PDE2AHSD11B1ALDH1A1LMNAKDM4E
SCHEMBL27185622 0.75 STING1 (0.60) PDE2AHSD11B1PDE10APDE3AKDM4E
SCHEMBL15187435 0.74 MARK3 (0.46) PDE2AHSD11B1PDE10APDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017108723-A2 PYRAZOLO[1,5a]PYRIMIDINE DERIVATIVES AS IRAK4 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2017-06-29 WO disclosed