SCHEMBL19050263

SCHEMBL19050263

O=C(O)c1cn(C[C@H](F)CO)nn1

nearest known ligand 0.43

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.43
GLS O94925 15/20 0.43
GRM2 Q14416 1/20 0.36
CA5A P35218 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19021038 0.86 DPP4 (0.42) DPP4GLSCA5A
SCHEMBL31124067 0.85 DPP4 (0.49) DPP4GLSGRM2CA5A
SCHEMBL17396743 0.80 GLS (0.43) DPP4GLS
SCHEMBL17396732 0.80 GLS (0.43) DPP4GLS
SCHEMBL29224209 0.79 DPP4 (0.42) DPP4GLSGRM2CA5A
SCHEMBL17396812 0.79 GLS (0.39) GLS
SCHEMBL17389096 0.79 GLS (0.39) GLS
SCHEMBL22062686 0.78 DPP4 (0.46) DPP4GLSCA5A
SCHEMBL4780340 0.77 DPP4 (0.42) DPP4GLSCA5A
SCHEMBL19050259 0.76 GLS (0.39) DPP4GLS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017112831-A1 SALT FORMS AND POLYMORPHS OF (R)-1-(4-(6-(2-(4-(3,3-DIFLUOROCYCLOBUTOXY)-6-METHYLPYRIDIN-2-YL) ACETAMIDO) PYRIDAZIN-3-YL)-2-FLUOROBUTYL)-N-METHYL-1H-1,2,3-TRIAZOLE-4-CARBOXAMIDE BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2017-06-29 WO disclosed