SCHEMBL1905475

SCHEMBL1905475

CCC1Cc2ccc(OC)cc2CCN1C(=O)C(F)(F)F

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.59
ESR2 Q92731 1/20 0.59
ABHD6 Q9BV23 1/20 0.46
KDM4E B2RXH2 2/20 0.44
LMNA P02545 2/20 0.44
ALDH1A1 P00352 1/20 0.44
MTNR1B P49286 4/20 0.43
HSD11B1 P28845 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
MAPT P10636 1/20 0.42
HTT P42858 1/20 0.42
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
DRD1 P21728 3/20 0.42
DRD5 P21918 3/20 0.42
DRD2 P14416 3/20 0.42
DRD3 P35462 3/20 0.42
DRD4 P21917 1/20 0.41
MTNR1A P48039 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2365603 0.82 ESR1 (0.59) ESR1ESR2ABHD6KDM4ELMNA
SCHEMBL13846949 0.81 GRIN2C (0.53) MTNR1BDRD1DRD5DRD2DRD3
SCHEMBL6631355 0.80 MTNR1B (0.46) ESR1ESR2LMNAMTNR1BHTT
SCHEMBL2309023 0.79 ESR1 (0.85) ESR1ESR2ABHD6HDAC1HDAC6
SCHEMBL18408493 0.78 MTNR1B (0.44) MTNR1BDRD1DRD5DRD2DRD3
SCHEMBL30878525 0.76 ESR1 (0.57) ESR1ESR2KDM4ELMNAALDH1A1
SCHEMBL30878562 0.76 ESR1 (0.57) ESR1ESR2KDM4ELMNAALDH1A1
SCHEMBL25722286 0.76 ESR1 (0.57) ESR1ESR2KDM4ELMNAALDH1A1
SCHEMBL1904807 0.75 ESR1 (0.50) ESR1ESR2MAPTDRD2DRD4
SCHEMBL3895230 0.74 ESR1 (1.00) ESR1ESR2ABHD6HDAC6DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2322162-A1 5HT2C receptor modulator compositions and methods of use Arena Pharmaceuticals, Inc. (US) 2011-05-18 EP disclosed