SCHEMBL19059202

SCHEMBL19059202

COc1ccc(CC(=O)N2CCC2)cc1F

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.60
GFER P55789 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.52
ALDH1A1 P00352 3/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
ATM Q13315 1/20 0.52
KDM4E B2RXH2 1/20 0.50
HPGD P15428 1/20 0.50
HSD17B10 Q99714 1/20 0.50
POLB P06746 1/20 0.49
MAPT P10636 1/20 0.48
KDM1A O60341 2/20 0.48
KCNH2 Q12809 1/20 0.48
PKM P14618 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2762440 0.84 HTT (0.52) HTTGFERSMN1; SMN2ALDH1A1MEN1
SCHEMBL22813664 0.84 KMT2A (0.52) ALDH1A1KMT2A
SCHEMBL17572090 0.82 HTT (0.61) HTTGFERSMN1; SMN2ALDH1A1MEN1
SCHEMBL19423896 0.81 HTT (0.60) HTTGFERSMN1; SMN2ALDH1A1MEN1
SCHEMBL19356243 0.81 HTT (0.60) HTTGFERSMN1; SMN2ALDH1A1MEN1
SCHEMBL12988833 0.80 ECE2 (0.51) HTTSMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL17572088 0.79 HTT (0.61) HTTGFERSMN1; SMN2ALDH1A1MEN1
SCHEMBL23095882 0.78 HTT (0.57) HTTGFERSMN1; SMN2ALDH1A1MEN1
SCHEMBL19419479 0.78 HTT (0.57) HTTGFERSMN1; SMN2ALDH1A1MEN1
SCHEMBL11304999 0.78 HTT (0.60) HTTGFERSMN1; SMN2ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2693882-B1 SUBSTITUTED CYCLOPROPYL COMPOUNDS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF TREATMENT MERCK SHARP & DOHME (US) 2017-06-28 EP disclosed