SCHEMBL19059382

SCHEMBL19059382

CCCCCC(C)(CCCCC)c1ccncc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 2/20 0.39
CNR2 P34972 3/20 0.38
CNR1 P21554 2/20 0.38
NAAA Q02083 1/20 0.38
KIF11 P52732 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
NPC1 O15118 2/20 0.34
LMNA P02545 2/20 0.34
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
ESR1 P03372 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24475344 0.98 CNR2 (0.40) CYP3A4CYP2D6CNR2CNR1NAAA
SCHEMBL19223950 0.98 CNR2 (0.40) CYP3A4CYP2D6CNR2CNR1NAAA
SCHEMBL19274594 0.98 CYP3A4 (0.38) CYP3A4CYP2D6CNR2CNR1NAAA
SCHEMBL24871939 0.98 CNR2 (0.40) CYP3A4CYP2D6CNR2CNR1NAAA
SCHEMBL21470858 0.96 CNR2 (0.40) CYP3A4CYP2D6CNR2CNR1NAAA
SCHEMBL21185893 0.96 ESR1 (0.39) CYP3A4CYP2D6CNR2CNR1NAAA
SCHEMBL18852691 0.96 CNR2 (0.40) CYP3A4CYP2D6CNR2CNR1NAAA
SCHEMBL21695082 0.94 CNR2 (0.39) CYP3A4CYP2D6CNR2CNR1NAAA
SCHEMBL19440675 0.94 CYP3A4 (0.40) CYP3A4CYP2D6CNR2CNR1NAAA
SCHEMBL19059539 0.92 CYP3A4 (0.37) CYP3A4CYP2D6CNR2CNR1NAAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200197524-A1 QUATERNIZED NICOTINAMIDE ADENINE DINUCLEOTIDE SALVAGE PATHWAY INHIBITOR CONJUGATES SEATTLE GENETICS, INC. (US) 2020-06-25 US disclosed
US-10011573-B2 Human androgen receptor DNA-binding domain (DBD) compounds as therapeutics and methods for their use THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2018-07-03 US disclosed
US-20170183319-A1 HUMAN ANDROGEN RECEPTOR DNA-BINDING DOMAN (DBD) COMPOUNDS AS THERAPEUTICS AND METHODS FOR THEIR USE THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2017-06-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200197524-A1 QUATERNIZED NICOTINAMIDE ADENINE DINUCLEOTIDE SALVAGE PATHWAY INHIBITOR CONJUGATES NAMPT, NNMT, NADK CYP3A4 4804/4885CYP2D6 4394/4885CNR2 1527/4885
US-10011573-B2 Human androgen receptor DNA-binding domain (DBD) compounds as therapeutics and methods for their use AR, SHBG, BRCA1 CYP3A4 1211/4885CYP2D6 464/4885CNR2 1300/4885
US-20170183319-A1 HUMAN ANDROGEN RECEPTOR DNA-BINDING DOMAN (DBD) COMPOUNDS AS THERAPEUTICS AND METHODS FOR THEIR USE AR, FSHR, ESRRB CYP3A4 1950/4885CYP2D6 703/4885CNR2 1512/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.