SCHEMBL1906249

SCHEMBL1906249

Cc1ccc(C(=O)N(c2ccccc2)C2CC2)cc1NC(=O)c1ccc(OCc2ccc(OCCN(C)C)cn2)cc1

nearest known ligand 0.48

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 15/20 0.48
SMO Q99835 14/20 0.48
CACNA1H O95180 2/20 0.43
CACNA1B Q00975 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL243273 0.84 MAPK14 (0.48) MAPK14SMO
SCHEMBL243811 0.76 MAPK14 (0.52) MAPK14SMO
SCHEMBL243760 0.72 MAPK14 (0.56) MAPK14SMO
SCHEMBL2904915 0.72 MAPK14 (0.52) MAPK14SMO
SCHEMBL243467 0.71 MAPK14 (0.50) MAPK14SMO
SCHEMBL1901397 0.71 MAPK14 (0.53) MAPK14SMO
SCHEMBL243419 0.70 MAPK14 (0.54) MAPK14SMO
SCHEMBL244357 0.70 MAPK14 (0.52) MAPK14SMO
Bromide SCHEMBL241935 0.70 MAPK14 (0.52) MAPK14SMO
SCHEMBL3649540 0.70 SMO (0.77) MAPK14SMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7943776-B2 Amide derivatives bearing a cyclopropylaminoacarbonyl substituent useful as cytokine inhibitors ASRAZENECA AB (SE) 2011-05-17 US disclosed
US-20070135440-A1 Amide derivatives bearing a cyclopropylaminoacarbonyl substituent useful as cytokine inhibitors ASTRAZENECA AB (SE) 2007-06-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070135440-A1 Amide derivatives bearing a cyclopropylaminoacarbonyl substituent useful as cytokine inhibitors IL2, IL6, IL1B MAPK14 1549/4885SMO 2872/4885CACNA1H 4080/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.