SCHEMBL19065281

SCHEMBL19065281

COC(=O)CCc1ccc(O)c(CO)n1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
KDM4E B2RXH2 3/20 0.46
HSD17B10 Q99714 2/20 0.41
HPGD P15428 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
LMNA P02545 2/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
KMT2A Q03164 1/20 0.39
EGFR P00533 2/20 0.38
HIF1A Q16665 1/20 0.38
RPS6KB2 Q9UBS0 1/20 0.36
MIF P14174 1/20 0.36
TSHR P16473 2/20 0.36
CYP4F2 P78329 1/20 0.36
CYP4A11 Q02928 1/20 0.36
GAA P10253 1/20 0.36
GFER P55789 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19079049 0.85 KDM4E (0.41) ALDH1A1KDM4EHSD17B10HPGDSMN1; SMN2
SCHEMBL8825474 0.84 KDM4E (0.45) ALDH1A1KDM4EHSD17B10HPGDSMN1; SMN2
SCHEMBL19088171 0.82 KDM4E (0.46) ALDH1A1KDM4ESMN1; SMN2LMNAKMT2A
SCHEMBL8825211 0.79 CYP4F2 (0.49) ALDH1A1KDM4EHSD17B10HPGDSMN1; SMN2
SCHEMBL415443 0.78 KDM4E (0.47) ALDH1A1KDM4EHSD17B10HPGDSMN1; SMN2
SCHEMBL8825405 0.77 HPGD (0.50) ALDH1A1KDM4EHSD17B10HPGDMAPT
SCHEMBL8825192 0.76 KDM4E (0.49) ALDH1A1KDM4EHSD17B10HPGDSMN1; SMN2
SCHEMBL8825306 0.75 KDM4E (0.48) ALDH1A1KDM4EHSD17B10HPGDSMN1; SMN2
SCHEMBL18981803 0.75 HPGD (0.44) ALDH1A1KDM4EHSD17B10HPGDSMN1; SMN2
SCHEMBL2854918 0.75 KDM4E (0.45) ALDH1A1KDM4EHSD17B10HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108541302-B Urea-based Prostate Specific Membrane Antigen (PSMA) inhibitors for imaging and therapy 五一一制药股份有限公司 2023-02-14 CN disclosed
EP-3397968-B1 UREA-BASED PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) INHIBITORS FOR IMAGING AND THERAPY FIVE ELEVEN PHARMA INC (US) 2021-09-29 EP disclosed
EP-3397968-B1 UREA-BASED PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) INHIBITORS FOR IMAGING AND THERAPY FIVE ELEVEN PHARMA INC (US) 2021-09-29 EP disclosed
US-10688200-B2 Urea-based prostate specific membrane antigen (PSMA) inhibitors for imaging and therapy FIVE ELEVEN PHARMA INC. (US) 2020-06-23 US disclosed
US-10688200-B2 Urea-based prostate specific membrane antigen (PSMA) inhibitors for imaging and therapy FIVE ELEVEN PHARMA INC. (US) 2020-06-23 US disclosed
EP-3397968-A1 UREA-BASED PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) INHIBITORS FOR IMAGING AND THERAPY Five Eleven Pharma Inc. (US) 2018-11-07 EP disclosed
WO-2017116994-A1 UREA-BASED PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) INHIBITORS FOR IMAGING AND THERAPY FIVE ELEVEN PHARMA INC. (US) 2017-07-06 WO disclosed
WO-2017116994-A1 UREA-BASED PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) INHIBITORS FOR IMAGING AND THERAPY FIVE ELEVEN PHARMA INC. (US) 2017-07-06 WO disclosed
US-20170189568-A1 UREA-BASED PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) INHIBITORS FOR IMAGING AND THERAPY FIVE ELEVEN PHARMA INC. 2017-07-06 US disclosed
US-20170189568-A1 UREA-BASED PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) INHIBITORS FOR IMAGING AND THERAPY FIVE ELEVEN PHARMA INC. 2017-07-06 US disclosed
US-20170189568-A1 UREA-BASED PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) INHIBITORS FOR IMAGING AND THERAPY FIVE ELEVEN PHARMA INC. 2017-07-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170189568-A1 UREA-BASED PROSTATE SPECIFIC MEMBRANE ANTIGEN (PSMA) INHIBITORS FOR IMAGING AND THERAPY KLK3, FOLH1, UTS2R ALDH1A1 1860/4885KDM4E 1861/4885HSD17B10 3608/4885
US-10688200-B2 Urea-based prostate specific membrane antigen (PSMA) inhibitors for imaging and therapy KLK3, FOLH1, UTS2R ALDH1A1 1860/4885KDM4E 1861/4885HSD17B10 3608/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.