SCHEMBL19082541

SCHEMBL19082541

CN1Cc2nccc(F)c2C1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.30
RAF1 P04049 1/20 0.30
RPS6KB1 P23443 1/20 0.30
MAPK1 P28482 1/20 0.30
AKT1 P31749 1/20 0.30
AKT2 P31751 1/20 0.30
KDR P35968 1/20 0.30
MAPKAPK2 P49137 1/20 0.30
PRKAG1 P54619 1/20 0.30
MAP2K1 Q02750 1/20 0.30
PRKAA1 Q13131 1/20 0.30
NEK1 Q96PY6 1/20 0.30
PRKAB1 Q9Y478 1/20 0.30
CSNK1D P48730 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19080438 0.78 HTR2C (0.33)
SCHEMBL22652449 0.78 KCNH2 (0.31)
SCHEMBL20652027 0.78 KCNH2 (0.31)
SCHEMBL19082532 0.76 HRH4 (0.36) IKBKBRAF1RPS6KB1MAPK1AKT1
SCHEMBL12853675 0.75 SLC6A2 (0.37)
SCHEMBL17624436 0.73 ROCK2 (0.34) IKBKBRAF1RPS6KB1MAPK1AKT1
SCHEMBL17624438 0.73 HTR2A (0.41)
SCHEMBL20651751 0.72 KCNH2 (0.36)
SCHEMBL256364 0.70 IKBKB (0.34) IKBKBRAF1RPS6KB1MAPK1AKT1
SCHEMBL17624435 0.70 UGCG (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020227368-A1 HSP90 INHIBITORS AND USES THEREOF TRUSTEES OF BOSTON UNIVERSITY (US) 2020-11-12 WO disclosed
WO-2017117447-A1 MULTICYCLIC COMPOUNDS AND USES THEREOF Karyopharm Therapeutics Inc. (US) 2017-07-06 WO disclosed