SCHEMBL19082532

SCHEMBL19082532

CN1Cc2nccc(N)c2C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
SLC6A2 P23975 4/20 0.35
SLC6A4 P31645 4/20 0.35
SLC6A3 Q01959 4/20 0.35
MAPK1 P28482 2/20 0.35
RGS12 O14924 1/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
ALOX12 P18054 1/20 0.35
NFKB1 P19838 1/20 0.35
HTR2A P28223 1/20 0.35
ADRA1A P35348 1/20 0.35
PTGS2 P35354 1/20 0.35
HRH1 P35367 1/20 0.35
OPRM1 P35372 1/20 0.35
GNAI1 P63096 1/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20651752 0.78 MITF (0.31) LMNA
SCHEMBL19079905 0.78 RAD52 (0.32)
SCHEMBL17624447 0.78 CCR1 (0.35) HRH4HRH3SLC6A2SLC6A4SLC6A3
SCHEMBL19082541 0.76 IKBKB (0.30) MAPK1IKBKBRAF1RPS6KB1AKT1
SCHEMBL4825313 0.75 SLC6A2 (0.42) SLC6A2SLC6A4SLC6A3MAPK1RGS12
SCHEMBL17624436 0.73 ROCK2 (0.34) HRH3MAPK1CYP1A2CYP3A4IKBKB
SCHEMBL17624438 0.73 HTR2A (0.41) SLC6A2SLC6A4SLC6A3CYP1A2CYP3A4
SCHEMBL20652026 0.73 DPP8 (0.33)
SCHEMBL256364 0.70 IKBKB (0.34) MAPK1IKBKBRAF1RPS6KB1AKT1
SCHEMBL6845547 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017117447-A1 MULTICYCLIC COMPOUNDS AND USES THEREOF Karyopharm Therapeutics Inc. (US) 2017-07-06 WO disclosed