SCHEMBL19084253

SCHEMBL19084253

COc1ccnc(C(=O)N[C@H]2CCCC[C@@H](CC(C)C)[C@H](C)OC2=O)c1O

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 4/20 0.35
TAS1R1 Q7RTX1 4/20 0.35
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
ADORA2A P29274 1/20 0.33
TAS1R2 Q8TE23 2/20 0.33
PDE10A Q9Y233 1/20 0.32
BRD4 O60885 1/20 0.32
HCRTR1 O43613 2/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
AXL P30530 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19084190 0.92 TAS1R3 (0.35) TAS1R3TAS1R1NPC1RAB9AADORA2A
SCHEMBL19084243 0.90 TAS1R3 (0.37) TAS1R3TAS1R1NPC1RAB9AADORA2A
SCHEMBL19088919 0.89 PDE4D (0.34) TAS1R3TAS1R1TAS1R2PDE10A
SCHEMBL19084225 0.88 NPC1 (0.32) NPC1RAB9AADORA2APDE10ABRD4
SCHEMBL19084186 0.88 TAS1R3 (0.35) TAS1R3TAS1R1NPC1RAB9AADORA2A
SCHEMBL19099682 0.86 TAS1R3 (0.34) TAS1R3TAS1R1NPC1RAB9AADORA2A
SCHEMBL19084210 0.86 TAS1R3 (0.38) TAS1R3TAS1R1NPC1RAB9AADORA2A
SCHEMBL19084260 0.86 NPC1 (0.31) NPC1RAB9AADORA2APDE10ABRD4
SCHEMBL17245180 0.86 TAS1R3 (0.32) TAS1R3TAS1R1NPC1RAB9AADORA2A
SCHEMBL16605181 0.85 TAS1R3 (0.33) TAS1R3TAS1R1NPC1RAB9AADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017116956-A1 MACROCYCLIC PICOLINAMIDES AS FUNGICIDES DOW AGROSCIENCES LLC (US) 2017-07-06 WO disclosed