SCHEMBL1908487

SCHEMBL1908487

CNC(=O)c1cn(C)c(=O)c2c(-c3ccccc3)c(-c3ccc(C4(N(C(=O)O)C(C)(C)C)CCC4)cc3)oc12

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 3/20 0.35
AKT2 P31751 3/20 0.35
BRD4 O60885 2/20 0.35
NR4A2 P43354 1/20 0.34
TNK2 Q07912 1/20 0.32
OPRM1 P35372 1/20 0.31
OPRL1 P41146 1/20 0.31
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1903884 0.91 AKT2 (0.33) AKT1AKT2BRD4OPRM1OPRL1
SCHEMBL1902498 0.90 OPRM1 (0.36) AKT1AKT2BRD4OPRM1OPRL1
SCHEMBL1905091 0.87
SCHEMBL12095384 0.84 AKT1 (0.48) AKT1AKT2BRD4NR4A2
SCHEMBL1904285 0.84 OPRL1 (0.32) TNK2OPRM1OPRL1
SCHEMBL1905277 0.82 BRD4 (0.38) AKT1AKT2BRD4NR4A2TNK2
SCHEMBL1907424 0.81 MEN1 (0.31) TNK2
SCHEMBL1903889 0.79 KDM4E (0.30) OPRM1KCNH2
SCHEMBL1907422 0.78 KDM4E (0.30) OPRM1KCNH2
SCHEMBL1904227 0.77 LCK (0.30) TNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011055115-A1 AKT / PKB INHIBITORS ALMAC DISCOVERY LIMITED (GB) 2011-05-12 WO disclosed