SCHEMBL19086018

SCHEMBL19086018

CC[C@@H](NC(=O)c1ccc2[nH]ncc2c1)C(=O)N1CCc2sc(C(=O)NC3CCOC3)cc2C1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 8/20 0.44
ROCK1 Q13464 3/20 0.44
MAPK14 Q16539 1/20 0.37
HDAC6 Q9UBN7 2/20 0.36
NAMPT P43490 5/20 0.36
CYP3A4 P08684 1/20 0.35
METTL3 Q86U44 1/20 0.35
KMT2A Q03164 1/20 0.35
AKT1 P31749 1/20 0.34
P2RY12 Q9H244 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086049 0.96 ROCK2 (0.43) ROCK2ROCK1MAPK14HDAC6CYP3A4
SCHEMBL19086054 0.94 ROCK2 (0.41) ROCK2ROCK1MAPK14HDAC6CYP3A4
SCHEMBL19086141 0.91 ROCK2 (0.44) ROCK2ROCK1MAPK14HDAC6CYP3A4
SCHEMBL19086020 0.91 ROCK2 (0.44) ROCK2ROCK1MAPK14HDAC6CYP3A4
SCHEMBL19086047 0.90 ROCK2 (0.44) ROCK2ROCK1MAPK14HDAC6CYP3A4
SCHEMBL19086052 0.90 ROCK2 (0.46) ROCK2ROCK1MAPK14HDAC6CYP3A4
SCHEMBL19086056 0.90 ROCK2 (0.43) ROCK2ROCK1MAPK14HDAC6CYP3A4
SCHEMBL19086051 0.89 ROCK2 (0.48) ROCK2ROCK1MAPK14HDAC6CYP3A4
SCHEMBL19086046 0.88 ROCK2 (0.41) ROCK2ROCK1MAPK14HDAC6CYP3A4
SCHEMBL19086050 0.88 ROCK2 (0.41) ROCK2ROCK1MAPK14HDAC6CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed