SCHEMBL19086025

SCHEMBL19086025

CNC(=O)c1cc2c(s1)CCN(C(=O)[C@H](NC(=O)c1ccc3[nH]ncc3c1)C(C)C)C2

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 8/20 0.43
HDAC6 Q9UBN7 3/20 0.39
ROCK2 O75116 5/20 0.39
CYP3A4 P08684 3/20 0.39
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
METTL3 Q86U44 1/20 0.37
PRMT5 O14744 1/20 0.37
WDR77 Q9BQA1 1/20 0.37
CCR1 P32246 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086161 0.92 HDAC6 (0.41) HDAC6ROCK2CYP3A4METTL3PRMT5
SCHEMBL19086156 0.88 HDAC6 (0.41) ENPP2HDAC6ROCK2CYP3A4METTL3
SCHEMBL19086154 0.86 F10 (0.43) HDAC6ROCK2CYP3A4PRMT5WDR77
SCHEMBL19086148 0.86 HDAC6 (0.40) HDAC6ROCK2CYP3A4METTL3PRMT5
SCHEMBL19086149 0.86 ANPEP (0.40) HDAC6ROCK2METTL3PRMT5WDR77
SCHEMBL19086153 0.85 KMT2A (0.49) ROCK2CYP3A4PRMT5WDR77
SCHEMBL19086162 0.84 KMT2A (0.40) HDAC6ROCK2CYP3A4METTL3PRMT5
SCHEMBL19086155 0.84 HDAC6 (0.38) HDAC6ROCK2CYP3A4METTL3PRMT5
SCHEMBL19086026 0.82 METTL3 (0.44) HDAC6ROCK2METTL3PRMT5WDR77
SCHEMBL19086160 0.82 HDAC6 (0.38) HDAC6ROCK2CYP3A4METTL3PRMT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed