SCHEMBL19086191

SCHEMBL19086191

O=C(Nc1ccccc1)c1cc2c(s1)CCN(C(=O)OCc1ccccc1)C2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 12/20 0.48
SIGMAR1 Q99720 12/20 0.48
PRMT5 O14744 3/20 0.47
WDR77 Q9BQA1 3/20 0.47
MEN1 O00255 2/20 0.47
ALDH1A1 P00352 2/20 0.47
KMT2A Q03164 2/20 0.47
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
HPGD P15428 1/20 0.47
ALOX15 P16050 1/20 0.47
HSD17B10 Q99714 1/20 0.47
DHFR P00374 1/20 0.46
HDAC6 Q9UBN7 2/20 0.45
HTR1A P08908 2/20 0.44
ADRA2A P08913 2/20 0.44
ADRA2B P18089 2/20 0.44
HRH2 P25021 2/20 0.44
HTR2A P28223 2/20 0.44
HTR2C P28335 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19086983 0.87 TMEM97 (0.53) TMEM97SIGMAR1MEN1ALDH1A1KMT2A
SCHEMBL3441575 0.82 TMEM97 (0.52) TMEM97SIGMAR1MEN1ALDH1A1KMT2A
SCHEMBL19086176 0.81 KDM1A (0.51) PRMT5WDR77MEN1ALDH1A1KMT2A
SCHEMBL19086175 0.78 HDAC6 (0.47) PRMT5WDR77MEN1ALDH1A1KMT2A
SCHEMBL11175834 0.77 TMEM97 (0.53) TMEM97SIGMAR1ALDH1A1HPGDHTR1A
SCHEMBL19086350 0.76 MAPT (0.48) PRMT5WDR77MEN1ALDH1A1KMT2A
SCHEMBL11173780 0.75 TMEM97 (0.48) TMEM97SIGMAR1MEN1ALDH1A1KMT2A
SCHEMBL324228 0.73 TMEM97 (0.67) TMEM97SIGMAR1PRMT5WDR77MEN1
SCHEMBL28523456 0.73 HDAC6 (0.53) PRMT5WDR77MEN1ALDH1A1KMT2A
SCHEMBL28523454 0.73 HDAC6 (0.53) PRMT5WDR77MEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017114275-A1 COMPOUND FOR INHIBITING ROCK, PREPARATION METHOD AND USE OF SAME 成都先导药物开发有限公司 2017-07-06 WO disclosed