SCHEMBL19135652

SCHEMBL19135652

BC(B)(Oc1cc2n(c(=O)n1)CC(C)(C)N2CC)c1cccc(F)c1F

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 4/20 0.32
GRM5 P41594 1/20 0.32
PDE4A P27815 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19135609 0.89 GPR84 (0.31) GPR84PDE4A
SCHEMBL19135647 0.88 GRM5 (0.31) GPR84GRM5PDE4A
SCHEMBL19135691 0.87 GPR84 (0.32) GPR84GRM5PDE4A
SCHEMBL15900849 0.82 GPR84 (0.46) GPR84GRM5PDE4A
SCHEMBL15901268 0.80 GPR84 (0.38) GPR84GRM5PDE4A
SCHEMBL19135640 0.79 P2RX7 (0.33) GPR84PDE4A
SCHEMBL19135646 0.74 GPR84 (0.44) GPR84PDE4A
SCHEMBL19135649 0.74 P2RX7 (0.31) GPR84
SCHEMBL15901284 0.72 GPR84 (0.35) GPR84GRM5PDE4A
SCHEMBL15900767 0.70 GPR84 (0.46) GPR84GRM5PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9708330-B2 2,3-dihydroimidazol[1,2-C]pyrimidin-5(1-H)-one based ipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitors GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-07-18 US disclosed