SCHEMBL19156379

SCHEMBL19156379

CC(=O)[C@H]1CCC2C3CCC4CC(=O)CCC4(C)C3CCC21C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B10 O60218 4/20 1.00
AKR1B1 P15121 4/20 1.00
GPBAR1 Q8TDU6 2/20 1.00
CYP3A4 P08684 3/20 0.70
SHBG P04278 2/20 0.70
CYP19A1 P11511 2/20 0.70
NR3C1 P04150 1/20 0.70
PGR P06401 1/20 0.70
SERPINA6 P08185 1/20 0.70
NR3C2 P08235 1/20 0.70
AR P10275 1/20 0.70
HSD17B10 Q99714 1/20 0.70
MGAM O43451 1/20 0.70
GABRP O00591 4/20 0.63
GABRD O14764 4/20 0.63
GABRA1 P14867 4/20 0.63
GABRB1 P18505 4/20 0.63
GABRG2 P18507 4/20 0.63
GABRB3 P28472 4/20 0.63
GABRA5 P31644 4/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18373741 1.00 AKR1B10 (1.00) AKR1B10AKR1B1GPBAR1CYP3A4SHBG
SCHEMBL13487248 1.00 AKR1B10 (1.00) AKR1B10AKR1B1GPBAR1CYP3A4SHBG
SCHEMBL14007476 1.00 AKR1B10 (1.00) AKR1B10AKR1B1GPBAR1CYP3A4SHBG
SCHEMBL12242383 1.00 AKR1B10 (1.00) AKR1B10AKR1B1GPBAR1CYP3A4SHBG
SCHEMBL37778 1.00 AKR1B10 (1.00) AKR1B10AKR1B1GPBAR1CYP3A4SHBG
SCHEMBL23699767 1.00 AKR1B10 (1.00) AKR1B10AKR1B1GPBAR1CYP3A4SHBG
SCHEMBL17776486 1.00 AKR1B10 (1.00) AKR1B10AKR1B1GPBAR1CYP3A4SHBG
SCHEMBL12646116 1.00 AKR1B10 (1.00) AKR1B10AKR1B1GPBAR1CYP3A4SHBG
SCHEMBL675417 1.00 AKR1B10 (1.00) AKR1B10AKR1B1GPBAR1CYP3A4SHBG
SCHEMBL13988206 1.00 AKR1B10 (1.00) AKR1B10AKR1B1GPBAR1CYP3A4SHBG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2709631-B9 ANTAGONISTS OF CB1 RECEPTOR INSERM - INST NAT DE LA SANTÉ ET DE LA RECH MÉDICALE (FR) 2017-07-26 EP disclosed