SCHEMBL1918784

SCHEMBL1918784

O=C(O)c1ccc([N+](=O)[O-])cc1C1CC=CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
TDP1 Q9NUW8 2/20 0.54
CYP3A4 P08684 1/20 0.54
ALOX15 P16050 1/20 0.54
MAPT P10636 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
HSP90AA1 P07900 2/20 0.46
HTT P42858 2/20 0.45
GAPDH P04406 1/20 0.44
HSPA1A P0DMV8 1/20 0.44
HSPA8 P11142 1/20 0.44
CD44 P16070 1/20 0.44
MSN P26038 1/20 0.44
PTPN7 P35236 1/20 0.44
EZH2 Q15910 1/20 0.44
TP53 P04637 2/20 0.43
CTSV O60911 1/20 0.43
CTSL P07711 1/20 0.43
CHRNB4 P30926 2/20 0.43
CHRNA3 P32297 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22123315 0.88 ALDH1A1 (0.57) ALDH1A1TDP1CYP3A4ALOX15MAPT
SCHEMBL743844 0.78 POLB (0.49) ALDH1A1TDP1CYP3A4ALOX15MAPT
SCHEMBL10608165 0.76 HSP90AA1 (0.56) ALDH1A1TDP1CYP3A4ALOX15MAPT
SCHEMBL6363108 0.75 ALDH1A1 (0.54) ALDH1A1TDP1CYP3A4ALOX15MAPT
SCHEMBL28255849 0.75 HTT (0.53) ALDH1A1TDP1CYP3A4ALOX15MAPT
SCHEMBL260006 0.75 ALDH1A1 (0.70) ALDH1A1TDP1CYP3A4ALOX15MAPT
SCHEMBL29226874 0.74 MPO (0.47) ALDH1A1TDP1CYP3A4ALOX15MAPT
SCHEMBL29226876 0.74 MPO (0.47) ALDH1A1TDP1CYP3A4ALOX15MAPT
SCHEMBL30313782 0.74 KMT2A (0.58) ALDH1A1TDP1CYP3A4ALOX15SMN1; SMN2
SCHEMBL27527312 0.74 KMT2A (0.58) ALDH1A1TDP1CYP3A4ALOX15SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2326652-A1 NITRO DERIVATIVES OF FURASEMIDE AND THEIR USE AS DIURETICS Merck Sharp & Dohme Corp. (US) 2011-06-01 EP disclosed
WO-2010014516-A1 NITRO DERIVATIVES OF FURASEMIDE AND THEIR USE AS DIURETICS MERCK & CO., INC. (US) 2010-02-04 WO disclosed