SCHEMBL19198529

SCHEMBL19198529

CNc1cc(C)c(C)cc1C

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
ESR1 P03372 1/20 0.33
RAPGEF4 Q8WZA2 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP2C19 P33261 1/20 0.30
BCHE P06276 1/20 0.30
CES1 P23141 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20160730 0.94 ESR1 (0.35) ESR1RAPGEF4CYP1A2CYP2C19
SCHEMBL850793 0.78 ESR1 (0.30) ESR1
SCHEMBL19198539 0.78 HDAC1 (0.31) TSHRESR1RAPGEF4
SCHEMBL18619502 0.78 ESR1 (0.30) ESR1
SCHEMBL12656572 0.78 CD44 (0.42) CYP3A4MAPK1ESR1RAPGEF4
SCHEMBL2741245 0.78 ALDH1A1 (0.50) CYP3A4TSHRMAPK1ESR1CYP1A2
SCHEMBL19199535 0.78 POLB (0.32) CYP3A4TSHRMAPK1ESR1BCHE
SCHEMBL10072631 0.78 CYP3A4 (0.55) CYP3A4TSHRMAPK1CYP1A2
SCHEMBL21760184 0.78 ESR1 (0.30) ESR1
SCHEMBL10072636 0.78 CYP3A4 (0.55) CYP3A4TSHRMAPK1ESR1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4393924-A1 IMIDAZO [1,2-A] PYRAZINE OR PYRAZOLO [1,5-A] PYRIMIDINE DERIVATIVE AND USE THEREOF Tencent Technology (Shenzhen) Company Limited (CN) 2024-07-03 EP disclosed
WO-2022087475-A1 REVERSE TRANSCRIPTION OF POLYNUCLEOTIDES COMPRISING UNNATURAL NUCLEOTIDES THE SCRIPPS RESEARCH INSTITUTE (US) 2022-04-28 WO disclosed
US-20170217970-A1 NOVEL PYRAZOLO[3,4-d]PYRIMIDINE COMPOUND OR SALT THEREOF TAIHO PHARMACEUTICAL CO., LTD. (JP) 2017-08-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170217970-A1 NOVEL PYRAZOLO[3,4-d]PYRIMIDINE COMPOUND OR SALT THEREOF ERBB2, JAK2, ERBB4 CYP3A4 3077/4885TSHR 994/4885MAPK1 57/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.