SCHEMBL20160730

SCHEMBL20160730

CNc1cc(C)c(NC)cc1C

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.35
RAPGEF4 Q8WZA2 2/20 0.33
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32
KDM4E B2RXH2 1/20 0.32
USP2 O75604 1/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
RECQL P46063 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HSD17B10 Q99714 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
NOS3 P29474 1/20 0.31
NOS2 P35228 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19198529 0.94 CYP3A4 (0.36) ESR1RAPGEF4CYP1A2CYP2C19
SCHEMBL10072631 0.84 CYP3A4 (0.55) CYP1A2KDM4EALDH1A1POLBMAPT
SCHEMBL850793 0.84 ESR1 (0.30) ESR1
SCHEMBL18619502 0.84 ESR1 (0.30) ESR1
SCHEMBL2741245 0.84 ALDH1A1 (0.50) ESR1CYP1A2CYP2C19KDM4EUSP2
SCHEMBL26288061 0.84 CYP3A4 (0.34) ESR1RAPGEF4KDM4EALDH1A1POLB
SCHEMBL12702757 0.80 MAPT (0.43) KDM4EALDH1A1POLBMAPTHSD17B10
SCHEMBL14367957 0.80 ALDH1A1 (0.33) ESR1RAPGEF4KDM4EALDH1A1POLB
SCHEMBL11017296 0.80 CD44 (0.44) ESR1CYP1A2KDM4EALDH1A1MAPT
SCHEMBL9230506 0.80 RAPGEF4 (0.32) ESR1RAPGEF4HSD17B10MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021127305-A1 METHODS AND COMPOSITIONS FOR INDUCING APOPTOSIS IN CANCER STEM CELLS VIRGINIA COMMONWEALTH UNIVERSITY (US) 2021-06-24 WO disclosed
WO-2018089967-A1 INHIBITORS OF CANCER INVASION, ATTACHMENT, AND/OR METASTASIS VIRGINIA COMMONWEALTH UNIVERSITY (US) 2018-05-17 WO disclosed