SCHEMBL19200481

SCHEMBL19200481

O=CNC1c2ccccc2C[C@@H]1NC(=O)C(c1ccc(F)cc1F)N1CC(F)C1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GRM7 Q14831 3/20 0.38
GHSR Q92847 4/20 0.38
PYGL P06737 2/20 0.35
OXTR P30559 7/20 0.35
CYP3A4 P08684 2/20 0.35
AVPR2 P30518 2/20 0.35
AVPR1A P37288 2/20 0.35
KCNH2 Q12809 1/20 0.33
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
MMP1 P03956 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19200271 0.85 GRM7 (0.41) GRM7GHSRPYGLOXTRCYP3A4
SCHEMBL19200400 0.85 GRM7 (0.41) GRM7GHSRPYGLOXTRCYP3A4
SCHEMBL19200269 0.84 KDM4D (0.42) GRM7GHSROXTRCYP3A4AVPR2
SCHEMBL20678653 0.83 GRM7 (0.41) GRM7PYGLOXTRCYP3A4AVPR2
SCHEMBL19200422 0.83 GRM7 (0.41) GRM7PYGLOXTRCYP3A4AVPR2
SCHEMBL20678656 0.83 GRM7 (0.41) GRM7PYGLOXTRCYP3A4AVPR2
SCHEMBL19200313 0.79 OXTR (0.40) GRM7GHSROXTRCYP3A4AVPR2
SCHEMBL19200952 0.76 KDM4D (0.41) GRM7GHSROXTRCYP3A4AVPR2
SCHEMBL19183091 0.76 KDM4D (0.41) GRM7GHSROXTRCYP3A4AVPR2
SCHEMBL19200374 0.75 KDM4D (0.40) GRM7GHSROXTRCYP3A4AVPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017131221-A1 INDANE DERIVATIVES AS MGLUR7 MODULATORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2017-08-03 WO disclosed