SCHEMBL1920235

SCHEMBL1920235

C/C(=C\c1ccc(C)cc1)C(=O)O

nearest known ligand 0.69

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 2/20 0.69
MAPT P10636 3/20 0.47
POLB P06746 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
TBXAS1 P24557 5/20 0.46
CYP2A6 P11509 1/20 0.44
FOS P01100 1/20 0.44
JUN P05412 1/20 0.44
TRPM8 Q7Z2W7 1/20 0.43
APEX1 P27695 1/20 0.43
ALDH1A1 P00352 3/20 0.43
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CYP3A4 P08684 1/20 0.43
HPGD P15428 1/20 0.43
GLA P06280 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL474138 1.00 AKR1C3 (0.69) AKR1C3MAPTPOLBNPC1RAB9A
SCHEMBL9956060 1.00 AKR1C3 (0.69) AKR1C3MAPTPOLBNPC1RAB9A
SCHEMBL4806412 0.94 AKR1C3 (0.62) AKR1C3MAPTPOLBNPC1RAB9A
SCHEMBL2462983 0.91 AKR1C3 (0.82) AKR1C3POLBTBXAS1APEX1ALDH1A1
SCHEMBL2462984 0.91 AKR1C3 (0.82) AKR1C3POLBTBXAS1APEX1ALDH1A1
SCHEMBL16353249 0.85 AKR1C3 (0.51) AKR1C3MAPTPOLBNPC1RAB9A
SCHEMBL2439316 0.84 AKR1C3 (0.48) AKR1C3MAPTPOLBNPC1RAB9A
SCHEMBL9609553 0.84 AKR1C3 (0.48) AKR1C3MAPTPOLBNPC1RAB9A
SCHEMBL30752457 0.84 AKR1C3 (0.48) AKR1C3MAPTPOLBNPC1RAB9A
SCHEMBL2439312 0.84 AKR1C3 (0.48) AKR1C3MAPTPOLBNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 67 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4121802-B1 HIGH REFRACTIVE INDEX SILOXANE INSERT MATERIALS FOR EMBEDDED CONTACT LENSES ALCON INC (CH) 2024-07-17 EP claimed
EP-3973934-B1 POLYCATIONIC POLYMER, COMPOSITION COMPRISING THE POLYCATIONIC POLYMER, AND PRODUCT, COMPRISING AN ACTIVE SURFACE, PROVIDED WITH THE POLYCATIONIC POLYMER COBATT (NL) 2023-12-20 EP claimed
EP-3728339-B1 COMPOSITION FOR OPHTHALMOLOGICAL PRODUCTS AMO Ireland (IE) 2022-07-06 EP claimed
EP-2303331-B1 OPHTHALMIC DEVICE HAVING THERAPEUTIC AGENT DELIVERY CAPABILITY AND METHOD OF FORMING SAME ALCON INC (CH) 2022-01-26 EP claimed
EP-3200840-B1 LOW-WATER CONTENT ACRYLATE-ACRYLAMIDE COPOLYMERS FOR OPHTHALMIC DEVICES ALCON INC (CH) 2021-11-17 EP claimed
EP-3200839-B1 HYDROPHOBIC ACRYLATE-ACRYLAMIDE COPOLYMERS FOR OPHTHALMIC DEVICES NOVARTIS AG (CH) 2019-09-04 EP claimed
EP-3223870-B1 WET-PACK INTRAOCULAR LENS MATERIALS WITH HIGH REFRACTIVE INDEX NOVARTIS AG (CH) 2018-09-26 EP claimed
EP-3326980-A1 HEAT RAY SHIELDING PARTICLE CONTAINING COMPOSITION AND HEAT RAY SHIELDING FILM Evonik Degussa GmbH (DE) 2018-05-30 EP claimed
EP-3077016-B1 SOFT ACRYLIC MATERIALS WITH HIGH REFRACTIVE INDEX AND MINIMIZED GLISTENING NOVARTIS AG (CH) 2018-05-16 EP claimed
EP-2292672-B1 Biocompatible polymers and co-polymers comprising amino acids in the side chain CIS PHARMA AG (CH) 2018-05-09 EP claimed
EP-1177227-B1 WATER PLASTICIZED HIGH REFRACTIVE INDEX POLYMER FOR OPHTHALMIC APPLICATIONS SURGIDEV CORP (US) 2003-10-01 EP claimed
EP-0914169-B1 MATERIALS FOR USE IN GLAUCOMA FILTRATION DEVICES ALCON LAB INC (US) 2003-07-30 EP claimed
EP-0851013-B1 Ink jet inks containing branched polymer dispersants and emulsion polymer additives DU PONT (US) 2003-05-28 EP claimed
EP-0851011-B1 Ink jet inks containing emulsion polymer additives stabilized with structured polymers DU PONT (US) 2002-05-22 EP claimed
EP-0518225-B2 Aqueous pigmented inks for ink jet printers DU PONT (US) 1999-10-20 EP claimed
EP-0633914-B1 An aqueous ink composition DU PONT (US) 1998-10-21 EP claimed
EP-0565709-B1 AQUEOUS INK JET INKS CONTAINING POLYOL/ALKYLENE OXIDE CONDENSATES AS COSOLVENTS DU PONT (US) 1996-11-13 EP claimed
EP-0509109-B1 Aqueous pigmented inks for ink jet printers DU PONT (US) 1995-07-12 EP claimed
EP-0633914-A1 PENETRANTS FOR AQUEOUS INK JET INKS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1995-01-18 EP claimed
WO-1992022614-A1 PENETRANTS FOR AQUEOUS INK JET INKS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1992-12-23 WO claimed