SCHEMBL19204853

SCHEMBL19204853

Cc1cc(F)c2[nH]nc(I)c2c1

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.32
ADORA2B P29275 1/20 0.32
CFTR P13569 1/20 0.31
MAPK1 P28482 1/20 0.30
MAP2K4 P45985 1/20 0.30
MAPKAPK2 P49137 1/20 0.30
MAPKAPK3 Q16644 1/20 0.30
MAPK6 Q16659 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29688902 0.82 MAPT (0.41) ADORA2AADORA2B
SCHEMBL5769361 0.82 MAPT (0.41) ADORA2AADORA2B
SCHEMBL13122336 0.81 ADORA2A (0.49) ADORA2AADORA2BCFTRMAPK1MAP2K4
SCHEMBL19249596 0.81 GPR84 (0.39)
SCHEMBL22890172 0.78 CHEK1 (0.34)
SCHEMBL19204854 0.78 AR (0.35)
SCHEMBL38661124 0.78 PDPK1 (0.31)
SCHEMBL31411446 0.77 TAAR1 (0.36) CFTRMAP2K4
SCHEMBL27221751 0.76 AR (0.35) ADORA2AADORA2B
SCHEMBL13122067 0.75 MAPK1 (0.34) ADORA2AADORA2BCFTRMAPK1MAP2K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017133667-A1 PYRIMIDINE AND PYRIDINE DERIVATIVES AND USE IN TREATMENT, AMELIORATION OR PREVENTION OF INFLUENZA THEREOF SAVIRA PHARMACEUTICALS GMBH (AT) 2017-08-10 WO disclosed
WO-2017133670-A1 PYRIDINE AND PYRIMIDINE DERIVATIVES AND THEIR USE IN TREATMENT, AMELIORATION OR PREVENTION OF INFLUENZA SAVIRA PHARMACEUTICALS GMBH (AT) 2017-08-10 WO disclosed