SCHEMBL19209583

SCHEMBL19209583

C#CCOc1cc(C(F)(F)F)nc2c(OC(F)(F)F)cccc12

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAOB P27338 10/20 0.39
SLC2A1 P11166 1/20 0.38
POLB P06746 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
LOXL2 Q9Y4K0 1/20 0.35
CYP3A4 P08684 1/20 0.34
CYP2A6 P11509 1/20 0.34
MAOA P21397 5/20 0.34
ALDH1A1 P00352 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
KDM4E B2RXH2 1/20 0.34
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
HSP90B1 P14625 1/20 0.34
KCNH2 Q12809 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19209590 0.78 MAOB (0.46) MAOBMAOAALDH1A1ADORA2AADORA1
SCHEMBL2859753 0.76 NPSR1 (0.43) POLBNPSR1ALDH1A1ADORA2AADORA1
SCHEMBL2849310 0.75 POLB (0.42) POLBNPSR1CYP3A4ALDH1A1ADORA2A
SCHEMBL3323333 0.72 MAOB (0.47) MAOBLOXL2CYP3A4CYP2A6MAOA
SCHEMBL26615234 0.71 CYP3A4 (0.43) MAOBLOXL2CYP3A4CYP2A6MAOA
SCHEMBL3952773 0.70 TNKS (0.47) NPSR1ALDH1A1ADORA2AKDM4E
SCHEMBL19209596 0.69 ACP1 (0.42) POLBNPSR1
SCHEMBL19209595 0.69 NPSR1 (0.38) POLBNPSR1ADORA2AADORA1KDM4E
SCHEMBL19209588 0.68 ALDH1A1 (0.35) SLC2A1LOXL2ALDH1A1KDM4E
SCHEMBL15473209 0.68 NPSR1 (0.44) SLC2A1NPSR1ALDH1A1KDM4EHSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017136642-A1 ANTIBIOTIC COMPOSITIONS THE TRUSTEES OF DARTMOUTH COLLEGE (US) 2017-08-10 WO disclosed
WO-2017136642-A1 ANTIBIOTIC COMPOSITIONS THE TRUSTEES OF DARTMOUTH COLLEGE (US) 2017-08-10 WO disclosed