SCHEMBL19209834

SCHEMBL19209834

CC(C)C(O)c1cc(Br)cnc1Cl

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
ALOX15 P16050 1/20 0.35
PPARG P37231 1/20 0.35
NCOA2 Q15596 1/20 0.35
NCOA1 Q15788 1/20 0.35
NCOA3 Q9Y6Q9 1/20 0.35
GABRA1 P14867 1/20 0.34
GABRB1 P18505 1/20 0.34
PLAU P00749 1/20 0.34
S1PR1 P21453 1/20 0.33
S1PR3 Q99500 1/20 0.33
MET P08581 1/20 0.32
PDE2A O00408 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2968350 0.85 GABRA1 (0.36) KMT2AMEN1TP53MAPTHPGD
SCHEMBL31254116 0.81 PLAU (0.32) KMT2AMEN1TP53MAPTHPGD
SCHEMBL20390070 0.81 GABRA1 (0.43) KMT2AMEN1TP53MAPTHPGD
SCHEMBL28634201 0.81 PLAU (0.33) KMT2AMEN1TP53MAPTHPGD
SCHEMBL28553372 0.79 S1PR1 (0.35) KMT2AMEN1TP53MAPTHPGD
SCHEMBL29555695 0.79 S1PR1 (0.35) KMT2AMEN1TP53MAPTHPGD
SCHEMBL24805816 0.79 PDE2A (0.38) PDE2A
SCHEMBL26587450 0.79 PDE2A (0.38) KMT2AGABRA1GABRB1METPDE2A
SCHEMBL27841463 0.77 KMT2A (0.37) KMT2AMEN1TP53MAPTHPGD
SCHEMBL18497256 0.75 ALDH1A1 (0.36) KMT2AMEN1TP53MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602799-B Kinase inhibitor 上海复尚慧创医药研究有限公司 2021-08-03 CN disclosed
WO-2017133701-A1 CERTAIN PROTEIN KINASE INHIBITORS SHANGHAI FOCHON PHARMACEUTICAL CO., LTD. (CN) 2017-08-10 WO disclosed