SCHEMBL19211158

SCHEMBL19211158

O=c1cc[nH]c2ccc(-c3ccccc3)cc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.58
NOTUM Q6P988 1/20 0.52
NR4A2 P43354 1/20 0.47
JAK2 O60674 1/20 0.45
ALDH1A1 P00352 3/20 0.44
CASP3 P42574 1/20 0.44
SENP7 Q9BQF6 1/20 0.44
SENP6 Q9GZR1 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
GLO1 Q04760 1/20 0.43
FEN1 P39748 1/20 0.43
TNKS2 Q9H2K2 1/20 0.42
MAP3K11 Q16584 1/20 0.42
MKNK1 Q9BUB5 1/20 0.41
HCRTR1 O43613 1/20 0.41
KDM4E B2RXH2 2/20 0.41
LMNA P02545 2/20 0.41
HPGD P15428 2/20 0.41
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19211220 0.84 TNKS2 (0.44) NPC1ALDH1A1MEN1KMT2ATNKS2
SCHEMBL19211223 0.83 ALDH1A1 (0.52) ALDH1A1MEN1KMT2ATNKS2KDM4E
Benzene SCHEMBL28794130 0.77 ALDH1A1 (0.53) ALDH1A1MEN1KMT2AKDM4ELMNA
SCHEMBL20667102 0.76 ADORA2A (0.53) NPC1JAK2MEN1KMT2AGLO1
SCHEMBL19211173 0.75 RHEB (0.53) NPC1KMT2ARAB9A
SCHEMBL10031 0.74 ALDH1A1 (0.55) ALDH1A1KMT2AKDM4ELMNAHPGD
SCHEMBL12338439 0.74 ALDH1A1 (0.65) NR4A2ALDH1A1KMT2AKDM4EHPGD
SCHEMBL28889107 0.74 NPC1 (0.66) NPC1NOTUMJAK2CASP3SENP7
SCHEMBL20657858 0.73 ALDH1A1 (0.44) NOTUMALDH1A1MEN1KMT2AHPGD
SCHEMBL1885355 0.73 ALDH1A1 (0.71) NPC1NR4A2ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3414229-A1 QUINOLINONE LYSYL OXIDASE-LIKE 2 INHIBITORS AND USES THEREOF Pharmakea, Inc. (US) 2018-12-19 EP disclosed
WO-2017139274-A1 QUINOLINONE LYSYL OXIDASE-LIKE 2 INHIBITORS AND USES THEREOF PHARMAKEA, INC. (US) 2017-08-17 WO disclosed