SCHEMBL1921244

SCHEMBL1921244

COC(=O)CNC(=O)c1cc(-c2ccc(Cl)cc2)ccn1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 9/20 0.61
EGLN3 Q9H6Z9 4/20 0.49
VEGFA P15692 3/20 0.49
FLT1 P17948 3/20 0.49
PSEN1 P49768 1/20 0.47
PSEN2 P49810 1/20 0.47
APH1B Q8WW43 1/20 0.47
NCSTN Q92542 1/20 0.47
APH1A Q96BI3 1/20 0.47
PSENEN Q9NZ42 1/20 0.47
MAPK1 P28482 1/20 0.47
MET P08581 1/20 0.44
ALDH1A1 P00352 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
NPSR1 Q6W5P4 1/20 0.43
MAPT P10636 1/20 0.43
MAP4K4 O95819 1/20 0.42
MMP13 P45452 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1921286 0.88 EGLN1 (0.60) EGLN1EGLN3VEGFAFLT1MAPK1
SCHEMBL1920884 0.87 EGLN1 (0.65) EGLN1EGLN3VEGFAFLT1MAPK1
SCHEMBL1921935 0.85 EGLN1 (0.70) EGLN1EGLN3VEGFAFLT1PSEN1
SCHEMBL27751614 0.85 LOXL2 (0.50) EGLN1EGLN3VEGFAFLT1MAPK1
SCHEMBL1921655 0.84 EGLN1 (0.65) EGLN1EGLN3VEGFAFLT1PSEN1
SCHEMBL12978818 0.84 EGLN1 (0.64) EGLN1EGLN3VEGFAFLT1MAPK1
SCHEMBL14319657 0.83 EGLN1 (0.56) EGLN1EGLN3PSEN1PSEN2APH1B
SCHEMBL1921195 0.81 EGLN1 (0.64) EGLN1EGLN3VEGFAFLT1ALDH1A1
SCHEMBL27751613 0.81 PSEN1 (0.46) EGLN1PSEN1PSEN2APH1BNCSTN
SCHEMBL20171252 0.80 EGLN1 (0.49) EGLN1EGLN3PSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 69 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044005-B8 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE WARNER CHILCOTT CO LLC (PR) 2012-12-05 EP claimed
EP-2044005-A2 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE The Procter and Gamble Company (US) 2009-04-08 EP claimed
WO-2008002576-A2 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE THE PROCTER & GAMBLE COMPANY (US) 2008-01-03 WO claimed
US-20070299086-A1 Prolyl hydroxylase inhibitors and methods of use THE PROCTER & GAMBLE COMPANY (US) 2007-12-27 US claimed
US-12478615-B2 Prolyl hydroxylase inhibitors and methods of use AKEBIA THERAPEUTICS, INC. (US) 2025-11-25 US disclosed
US-20240358691-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE WARNER CHILCOTT COMPANY, LLC (PR) 2024-10-31 US disclosed
US-11883386-B2 Prolyl hydroxylase inhibitors and methods of use AKEBIA THERAPEUTICS, INC. (US) 2024-01-30 US disclosed
US-20230201178-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE KREOS CAPITAL VII (UK) LIMITED (GB) 2023-06-29 US disclosed
US-20230201178-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE KREOS CAPITAL VII (UK) LIMITED (GB) 2023-06-29 US disclosed
EP-4095127-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE Akebia Therapeutics Inc. (US) 2022-11-30 EP disclosed
US-11426393-B2 Prolyl hydroxylase inhibitors and methods of use AKEBIA THERAPEUTICS, INC. (US) 2022-08-30 US disclosed
US-11426393-B2 Prolyl hydroxylase inhibitors and methods of use AKEBIA THERAPEUTICS, INC. (US) 2022-08-30 US disclosed
US-7811595-B2 such as {[5-(3-Chloro-phenyl)-3-hydroxy-pyridine-2-carbonyl]-amino}-acetic acid methyl ester; for controlling Peripheral Vascular Disease, Coronary Artery Disease, heart failure, ischemia, and anemia WARNER CHILCOTT COMPANY, LLC (US) 2010-10-12 US disclosed
US-7811595-B2 such as {[5-(3-Chloro-phenyl)-3-hydroxy-pyridine-2-carbonyl]-amino}-acetic acid methyl ester; for controlling Peripheral Vascular Disease, Coronary Artery Disease, heart failure, ischemia, and anemia WARNER CHILCOTT COMPANY, LLC (US) 2010-10-12 US disclosed
US-7811595-B2 such as {[5-(3-Chloro-phenyl)-3-hydroxy-pyridine-2-carbonyl]-amino}-acetic acid methyl ester; for controlling Peripheral Vascular Disease, Coronary Artery Disease, heart failure, ischemia, and anemia WARNER CHILCOTT COMPANY, LLC (US) 2010-10-12 US disclosed
EP-2044005-A2 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE The Procter and Gamble Company (US) 2009-04-08 EP disclosed
WO-2008002576-A2 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE THE PROCTER & GAMBLE COMPANY (US) 2008-01-03 WO disclosed
US-20070299086-A1 Prolyl hydroxylase inhibitors and methods of use THE PROCTER & GAMBLE COMPANY (US) 2007-12-27 US disclosed
US-20070299086-A1 Prolyl hydroxylase inhibitors and methods of use THE PROCTER & GAMBLE COMPANY (US) 2007-12-27 US disclosed
US-20070299086-A1 Prolyl hydroxylase inhibitors and methods of use THE PROCTER & GAMBLE COMPANY (US) 2007-12-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11426393-B2 Prolyl hydroxylase inhibitors and methods of use HIF1AN, EGLN3, HIF1A EGLN1 6/4885EGLN3 2/4885VEGFA 117/4885
US-11883386-B2 Prolyl hydroxylase inhibitors and methods of use HIF1AN, EGLN3, HIF1A EGLN1 6/4885EGLN3 2/4885VEGFA 117/4885
US-20240358691-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE HIF1AN, EGLN3, EGLN2 EGLN1 6/4885EGLN3 2/4885VEGFA 76/4885
US-12478615-B2 Prolyl hydroxylase inhibitors and methods of use HIF1AN, EGLN3, HIF1A EGLN1 6/4885EGLN3 2/4885VEGFA 117/4885
US-20230201178-A1 PROLYL HYDROXYLASE INHIBITORS AND METHODS OF USE HIF1AN, EGLN3, HIF1A EGLN1 6/4885EGLN3 2/4885VEGFA 117/4885
US-20070299086-A1 Prolyl hydroxylase inhibitors and methods of use HIF1AN, EGLN3, HIF1A EGLN1 6/4885EGLN3 2/4885VEGFA 117/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.