SCHEMBL19217038

SCHEMBL19217038

CS(=O)(=O)N1CCN(C(=O)c2cc3c(N4CC5COCC4C5)nc(-c4ccc(N)cc4)nn3c2)CC1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 10/20 0.43
PIK3R1 P27986 4/20 0.43
PIK3CD O00329 2/20 0.36
PIK3CB P42338 2/20 0.36
PIK3CG P48736 2/20 0.36
ACACB O00763 1/20 0.34
ACACA Q13085 1/20 0.34
MTOR P42345 3/20 0.33
EPHX2 P34913 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
MAPK1 P28482 1/20 0.33
SETD7 Q8WTS6 1/20 0.33
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19216914 0.85 PIK3CA (0.51) PIK3CAPIK3R1PIK3CDPIK3CBPIK3CG
SCHEMBL19217037 0.84 MAP3K12 (0.31) PIK3CAPIK3CGMTOR
SCHEMBL16611524 0.81 PIK3CA (0.60) PIK3CAPIK3R1PIK3CDPIK3CBPIK3CG
SCHEMBL16613103 0.80 PIK3CA (0.49) PIK3CAPIK3R1PIK3CDPIK3CBPIK3CG
SCHEMBL19217036 0.76 PIK3CA (0.44) PIK3CAPIK3R1PIK3CDPIK3CBPIK3CG
SCHEMBL16727864 0.71 PIK3CA (0.56) PIK3CAPIK3R1PIK3CDPIK3CBPIK3CG
SCHEMBL16727865 0.70 MTOR (0.47) PIK3CAPIK3R1PIK3CDMTOR
SCHEMBL19216996 0.68 PIK3CA (0.75) PIK3CAPIK3R1PIK3CDPIK3CBPIK3CG
SCHEMBL19216877 0.68 PIK3CA (0.59) PIK3CAPIK3R1PIK3CDPIK3CBPIK3CG
SCHEMBL16611585 0.67 PIK3CA (0.76) PIK3CAPIK3R1PIK3CDPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9724352-B2 Pyrrolo[2,1-F[1,2,4]triazine compounds, preparation methods and applications thereof SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES (CN) 2017-08-08 US disclosed