SCHEMBL19217036

SCHEMBL19217036

COC1CCCN(c2nc(-c3ccc(N)cc3)nn3cc(C(=O)N4CCN(S(C)(=O)=O)CC4)cc23)C1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 7/20 0.44
PIK3R1 P27986 1/20 0.44
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
MTOR P42345 2/20 0.35
CCNE1 P24864 1/20 0.35
CDK2 P24941 1/20 0.35
PIK3CD O00329 1/20 0.34
PIK3CB P42338 1/20 0.34
PIK3CG P48736 1/20 0.34
PARP1 P09874 2/20 0.34
PARP2 Q9UGN5 2/20 0.34
ACACB O00763 1/20 0.34
ACACA Q13085 1/20 0.34
ADRA1A P35348 1/20 0.34
DGAT2 Q96PD7 1/20 0.34
MAPK1 P28482 1/20 0.33
FFAR2 O15552 1/20 0.33
ADORA2A P29274 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19217040 0.85 ACACB (0.36) PIK3CAMTORPIK3CGPARP1PARP2
SCHEMBL19217039 0.84 ACACB (0.37) PIK3CAPIK3R1MTORPIK3CDPIK3CB
SCHEMBL16613103 0.84 PIK3CA (0.49) PIK3CAPIK3R1MTORCCNE1CDK2
SCHEMBL19216878 0.82 PIK3CA (0.56) PIK3CAPIK3R1MTORPIK3CDPIK3CB
SCHEMBL16611524 0.82 PIK3CA (0.60) PIK3CAPIK3R1MTORPIK3CDPIK3CB
SCHEMBL19217038 0.76 PIK3CA (0.43) PIK3CAPIK3R1ALDH1A1GAAMTOR
SCHEMBL16727865 0.74 MTOR (0.47) PIK3CAPIK3R1MTORPIK3CD
SCHEMBL19216983 0.74 ALKBH5 (0.37) ALDH1A1
SCHEMBL16727864 0.72 PIK3CA (0.56) PIK3CAPIK3R1MTORPIK3CDPIK3CB
SCHEMBL16613163 0.68 PIK3CA (0.68) PIK3CAPIK3R1MTORPIK3CDPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9724352-B2 Pyrrolo[2,1-F[1,2,4]triazine compounds, preparation methods and applications thereof SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES (CN) 2017-08-08 US disclosed