SCHEMBL19217042

SCHEMBL19217042

COC(=O)c1cc2c(N3CC4COC(C4)C3)nc(-c3ccc(N)cc3)nn2c1

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 8/20 0.34
PIK3CG P48736 2/20 0.34
PIK3R1 P27986 2/20 0.34
PIK3CD O00329 1/20 0.34
PIK3CB P42338 1/20 0.34
RAB9A P51151 2/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MTOR P42345 5/20 0.34
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAPK14 Q16539 2/20 0.32
CSNK1G1 Q9HCP0 1/20 0.32
TGFBR1 P36897 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16613162 0.87 MTOR (0.46) PIK3CAMTOR
SCHEMBL16610955 0.80 PIK3CA (0.49) PIK3CAPIK3CGPIK3R1PIK3CDPIK3CB
SCHEMBL19217039 0.77 ACACB (0.37) PIK3CAPIK3CGPIK3R1PIK3CDPIK3CB
SCHEMBL16613115 0.75 MTOR (0.48) PIK3CAMTOR
SCHEMBL16731005 0.75 MTOR (0.41) PIK3CAPIK3CBMTOR
SCHEMBL16613177 0.75 MTOR (0.41) PIK3CAPIK3CBMTOR
SCHEMBL16727865 0.71 MTOR (0.47) PIK3CAPIK3R1PIK3CDMTOR
SCHEMBL16727861 0.70 MTOR (0.51) PIK3CAPIK3R1ALDH1A1MTOR
SCHEMBL19217037 0.70 MAP3K12 (0.31) PIK3CAPIK3CGMTORMAPK14CSNK1G1
SCHEMBL19217040 0.69 ACACB (0.36) PIK3CAPIK3CGMTORMAPTMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9724352-B2 Pyrrolo[2,1-F[1,2,4]triazine compounds, preparation methods and applications thereof SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES (CN) 2017-08-08 US disclosed