SCHEMBL19217040

SCHEMBL19217040

COC1CCCN(c2nc(-c3ccc(N)cc3)nn3cc(C(=O)O)cc23)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 3/20 0.36
MAP4K4 O95819 1/20 0.36
FFAR2 O15552 1/20 0.36
EGLN1 Q9GZT9 1/20 0.35
PIK3CA P42336 1/20 0.35
MTOR P42345 1/20 0.35
PIK3CG P48736 1/20 0.35
MAPK14 Q16539 1/20 0.35
CSNK1G1 Q9HCP0 1/20 0.35
GSK3B P49841 2/20 0.35
GBA1 P04062 2/20 0.35
MAOB P27338 1/20 0.34
HTR6 P50406 1/20 0.34
PPARA Q07869 1/20 0.34
MAPT P10636 1/20 0.34
LRRK2 Q5S007 2/20 0.34
AVPR1B P47901 1/20 0.34
PARP1 P09874 1/20 0.33
PARP2 Q9UGN5 1/20 0.33
PDE4A P27815 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19217039 0.92 ACACB (0.37) ACACBMAP4K4FFAR2PIK3CAMTOR
SCHEMBL19217036 0.85 PIK3CA (0.44) ACACBFFAR2PIK3CAMTORPIK3CG
SCHEMBL19216983 0.80 ALKBH5 (0.37) PPARAMAPTAVPR1B
SCHEMBL16613115 0.79 MTOR (0.48) PIK3CAMTOR
SCHEMBL16611831 0.78 PIK3CA (0.48) EGLN1PIK3CAMTORPIK3CGMAPK14
SCHEMBL16613162 0.74 MTOR (0.46) PIK3CAMTOR
SCHEMBL16610955 0.72 PIK3CA (0.49) PIK3CAMTORPIK3CGMAPK14CSNK1G1
SCHEMBL19217037 0.70 MAP3K12 (0.31) PIK3CAMTORPIK3CGMAPK14CSNK1G1
SCHEMBL16727865 0.70 MTOR (0.47) PIK3CAMTOR
SCHEMBL19217042 0.69 PIK3CA (0.34) PIK3CAMTORPIK3CGMAPK14CSNK1G1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9724352-B2 Pyrrolo[2,1-F[1,2,4]triazine compounds, preparation methods and applications thereof SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES (CN) 2017-08-08 US disclosed