Fluphenazine

Fluphenazine

SCHEMBL19221

OCCN1CCN(CCCN2c3ccccc3Sc3ccc(C(F)(F)F)cc32)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

DRD2

The experimentally established mechanism targets of Fluphenazine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 known ✓ P14416 3/20 1.00
LMNA P02545 7/20 1.00
MAPT P10636 7/20 1.00
CYP3A4 P08684 5/20 1.00
MAPK1 P28482 5/20 1.00
USP2 O75604 5/20 1.00
TP53 P04637 4/20 1.00
ABCB11 O95342 3/20 1.00
CYP1A2 P05177 3/20 1.00
HTR1A P08908 3/20 1.00
ADRA2A P08913 3/20 1.00
CYP2D6 P10635 3/20 1.00
ADRA2B P18089 3/20 1.00
ADRA2C P18825 3/20 1.00
NFKB1 P19838 3/20 1.00
SLC6A2 P23975 3/20 1.00
HTR2A P28223 3/20 1.00
HTR2C P28335 3/20 1.00
SLC6A4 P31645 3/20 1.00
ADRA1A P35348 3/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fluphenazine SCHEMBL29354183 1.00 LMNA (1.00) LMNAMAPTCYP3A4MAPK1USP2
Fluphenazine SCHEMBL5072860 1.00 LMNA (1.00) LMNAMAPTCYP3A4MAPK1USP2
Fluphenazine SCHEMBL29388890 1.00 LMNA (1.00) LMNAMAPTCYP3A4MAPK1USP2
Fluphenazine SCHEMBL28642082 0.99 LMNA (0.98) LMNAMAPTCYP3A4MAPK1USP2
Fluphenazine SCHEMBL30390918 0.99 LMNA (1.00) LMNAMAPTCYP3A4MAPK1USP2
Fluphenazine SCHEMBL2560022 0.99 LMNA (1.00) LMNAMAPTCYP3A4MAPK1USP2
Fluphenazine SCHEMBL41634 0.99 LMNA (1.00) LMNAMAPTCYP3A4MAPK1USP2
Fluphenazine SCHEMBL29860638 0.99 LMNA (1.00) LMNAMAPTCYP3A4MAPK1USP2
Fluphenazine SCHEMBL7194252 0.99 LMNA (0.98) LMNAMAPTCYP3A4MAPK1USP2
Fluphenazine SCHEMBL41635 0.99 LMNA (1.00) LMNAMAPTCYP3A4MAPK1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 24953 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3607938-B1 PHARMACEUTICAL COMPOSITION SOVIC BRKICIC LJILJANA (HR) 2026-05-27 EP claimed
US-12624036-B2 Method of treating post-traumatic stress disorder INTRA-CELLULAR THERAPIES, INC. (US) 2026-05-12 US claimed
US-12624037-B2 Method of treating agitation, aggressive behavior, and impulse control disorder INTRA-CELLULAR THERAPIES, INC. (US) 2026-05-12 US claimed
CN-122028919-A Compositions and methods for treating cancer by affecting cancer cell membrane receptors and exosomes derived therefrom 黄奇英 2026-05-12 CN claimed
EP-4736841-A1 A MUCOADHESIVE LAYER FOR BUCCAL ADMINISTRATION OF AN ACTIVE PHARMACEUTICAL INGREDIENT IQ medical GmbH (DE) 2026-05-06 EP claimed
WO-2026090360-A1 FUSED PYRIMIDINE COMPOUNDS FOR TREATMENT OF TINNITUS, HEARING LOSS, AND MENIERE'S DISEASE OVID THERAPEUTICS INC. (US) 2026-04-30 WO claimed
US-20260108529-A1 FUSED AMINO PYRIMIDINE COMPOUNDS FOR TREATMENT OF TINNITUS, ACUTE SENSORINEURAL HEARING LOSS, AGE-RELATED HEARING LOSS, AND MENIERE'S DISEASE OVID THERAPEUTICS INC (US) 2026-04-23 US claimed
US-20260103758-A1 METHODS AND BIOMARKERS FOR TREATING BREAST CANCER KING ABDULAZIZ UNIVERSITY (SA) 2026-04-16 US claimed
EP-4724062-A2 COMPOSITIONS AND METHODS FOR INCREASING EXPOSURE OF R(-)-MDA EmpathBio, Inc. (US) 2026-04-15 EP claimed
US-12594388-B2 Device to deliver a predetermined amount of a substance to a natural orifice of the body APTARGROUP, INC. (US) 2026-04-07 US claimed
WO-1983000086-A1 USE OF CALMODULIN BINDING DRUGS IN UTERUS TO PREVENT PREGNANCY UNIV GEORGIA RES FOUND (US) 1983-01-20 WO claimed
US-4369172-A Prolonged release therapeutic compositions based on hydroxypropylmethylcellulose FOREST LABORATORIES INC. (US) 1983-01-18 US claimed
EP-0053108-A1 VAGINAL CONTRACEPTIVES COMPRISING PSYCHOACTIVE DRUGS THE UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 1982-06-09 EP claimed
WO-1981003421-A1 USE OF PSYCHOACTIVE DRUGS AS VAGINAL CONTRACEPTIVES UNIV GEORGIA (US) 1981-12-10 WO claimed
EP-0022771-A4 RADIO RECEPTOR ASSAY FOR BENZODIAZEPINES IN PLASMA AND OTHER BIOLOGICAL SPECIMENS. US HEALTH (US) 1981-02-04 EP claimed
EP-0022771-A1 RADIO RECEPTOR ASSAY FOR BENZODIAZEPINES IN PLASMA AND OTHER BIOLOGICAL SPECIMENS THE UNITED STATES OF AMERICA, represented by DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1981-01-28 EP claimed
WO-1980000750-A1 RADIO RECEPTOR ASSAY FOR BENZODIZAPINES IN PLASMA AND OTHER BIOLOGICAL SPECIMENS US COMMERCE (US) 1980-04-17 WO claimed
US-4197288-A Neuroleptic radioreceptor assay method and kit BURROUGHS WELLCOME CO. (US) 1980-04-08 US claimed
US-4175119-A Composition and method to prevent accidental and intentional overdosage with psychoactive drugs PORTER GARRY L 1979-11-20 US claimed
US-3993072-A Microporous drug delivery device ALZA CORPORATION (US) 1976-11-23 US claimed