SCHEMBL19225503

SCHEMBL19225503

CC(C#N)(COCc1ccccc1)NSC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.40
KDM4E B2RXH2 1/20 0.40
POLB P06746 1/20 0.40
SGMS2 Q8NHU3 1/20 0.39
MAOB P27338 1/20 0.37
CTSS P25774 3/20 0.37
CHRM3 P20309 3/20 0.36
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
OPRM1 P35372 1/20 0.35
DRD3 P35462 1/20 0.35
CTSL P07711 4/20 0.34
CTSB P07858 4/20 0.34
CTSK P43235 3/20 0.34
TACR1 P25103 1/20 0.34
ALDH1A1 P00352 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15776475 0.76 SGMS2 (0.37) TSHRKDM4EPOLBSGMS2MAOB
SCHEMBL3301730 0.76 TSHR (0.50) TSHRKDM4EPOLBSGMS2MAOB
SCHEMBL3338802 0.76 TSHR (0.50) TSHRKDM4EPOLBSGMS2MAOB
SCHEMBL19225502 0.75 CTSS (0.37) TSHRKDM4EPOLBSGMS2MAOB
SCHEMBL5529079 0.73 KDM4E (0.53) TSHRKDM4EPOLBSGMS2MAOB
SCHEMBL6043011 0.71 TSHR (0.58) TSHRKDM4EPOLBTACR1ALDH1A1
SCHEMBL20267540 0.70 TSHR (0.47) TSHRKDM4EPOLBSGMS2MAOB
SCHEMBL3474055 0.70 TSHR (0.56) TSHRKDM4EPOLBTACR1ALDH1A1
SCHEMBL19225650 0.70 KDM4E (0.42) TSHRKDM4EPOLBTACR1ALDH1A1
SCHEMBL1691827 0.69 TSHR (0.61) TSHRKDM4EPOLBTACR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2928867-B1 PYRIDINE-2-AMIDES USEFUL AS CB2 AGONISTS HOFFMANN LA ROCHE (CH) 2017-08-09 EP disclosed