SCHEMBL19225532

SCHEMBL19225532

O=C1C(Cc2c[nH]c3c(Cl)cccc23)NC(O)N1CCC#Cc1cnc2cccnn12

nearest known ligand 0.55

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 7/20 0.55
RIPK2 O43353 1/20 0.55
RIPK3 Q9Y572 1/20 0.55
TNF P01375 5/20 0.37
ABL1 P00519 3/20 0.31
CYP3A4 P08684 1/20 0.30
KCNH2 Q12809 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16084954 0.85 RIPK1 (0.70) RIPK1RIPK2RIPK3TNF
SCHEMBL16085003 0.84 RIPK1 (0.62) RIPK1RIPK2RIPK3TNF
SCHEMBL16084985 0.76 RIPK1 (0.63) RIPK1RIPK2RIPK3TNFABL1
SCHEMBL19225593 0.75 RIPK1 (0.48) RIPK1RIPK2RIPK3TNFABL1
SCHEMBL16084949 0.72 RIPK1 (0.79) RIPK1RIPK2RIPK3TNFABL1
SCHEMBL16084948 0.72 RIPK1 (0.79) RIPK1RIPK2RIPK3TNFABL1
SCHEMBL16084958 0.72 RIPK1 (0.92) RIPK1RIPK2RIPK3TNFABL1
SCHEMBL16084969 0.71 RIPK1 (0.75) RIPK1RIPK2RIPK3ABL1CYP3A4
SCHEMBL17471719 0.71 RIPK1 (0.99) RIPK1RIPK2RIPK3TNFABL1
SCHEMBL16084944 0.71 RIPK1 (0.90) RIPK1RIPK2RIPK3TNFABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9725452-B2 Substituted indoles and pyrroles as RIP kinase inhibitors PRESIDENTS AND FELLOWS OF HARVARD COLLEGE (US) 2017-08-08 US disclosed