SCHEMBL19230442

SCHEMBL19230442

CC(=O)[C@@H](Cc1ccc(F)cc1)N(C)C

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
OPRM1 P35372 1/20 0.43
OPRD1 P41143 1/20 0.43
OPRK1 P41145 1/20 0.43
TDP1 Q9NUW8 2/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
HTT P42858 1/20 0.41
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
RIPK1 Q13546 2/20 0.41
CPA1 P15085 1/20 0.41
POLB P06746 1/20 0.40
APEX1 P27695 1/20 0.40
TAAR1 Q96RJ0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19230448 1.00 TRPA1 (0.44) TRPA1MEN1KMT2AOPRM1OPRD1
SCHEMBL16743936 0.84 ESR1 (0.56) OPRM1OPRD1OPRK1ALDH1A1MAPT
SCHEMBL18747135 0.84 ESR1 (0.56) OPRM1OPRD1OPRK1ALDH1A1MAPT
SCHEMBL15778554 0.84 ALDH1A1 (0.43) MEN1KMT2AOPRM1OPRD1OPRK1
SCHEMBL684451 0.82 ALDH1A1 (0.45) MEN1KMT2AALDH1A1MAPTHTT
SCHEMBL4745249 0.82 ACACB (0.44) MEN1KMT2AOPRM1OPRD1ALDH1A1
SCHEMBL13323473 0.82 ALDH1A1 (0.45) MEN1KMT2AALDH1A1MAPTHTT
SCHEMBL12341937 0.81 ALDH1A1 (0.59) MEN1KMT2AALDH1A1MAPTHTT
SCHEMBL8605469 0.81 ALDH1A1 (0.59) MEN1KMT2AALDH1A1MAPTHTT
SCHEMBL890230 0.81 ALDH1A1 (0.59) MEN1KMT2AALDH1A1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017136708-A1 SYNTHESIS AND COMPOSITION OF RAPAFUCIN LIBRARIES THE JOHNS HOPKINS UNIVERSITY (US) 2017-08-10 WO disclosed