SCHEMBL19230445

SCHEMBL19230445

CC(=O)[C@H](Cc1cccc2ccccc12)N(C)C

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTNNB1 P35222 1/20 0.51
MMP9 P14780 1/20 0.50
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C19 P33261 1/20 0.49
TDP1 Q9NUW8 1/20 0.47
OPRM1 P35372 4/20 0.46
L3MBTL1 Q9Y468 1/20 0.43
OPRD1 P41143 1/20 0.43
MME P08473 2/20 0.43
ACE P12821 2/20 0.43
TACR1 P25103 1/20 0.43
ACP3 P15309 1/20 0.42
CPA1 P15085 1/20 0.42
ACE2 Q9BYF1 1/20 0.42
MTNR1A P48039 1/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19230443 1.00 CTNNB1 (0.51) CTNNB1MMP9CYP1A2CYP2D6CYP2C19
SCHEMBL7297662 0.81 CTNNB1 (0.46) CTNNB1MMP9CYP1A2CYP2D6CYP2C19
SCHEMBL16743938 0.79 CTNNB1 (0.55) CTNNB1MMP9TDP1L3MBTL1MME
SCHEMBL6623784 0.79 CTNNB1 (0.55) CTNNB1MMP9TDP1L3MBTL1MME
SCHEMBL13879137 0.79 CTNNB1 (0.55) CTNNB1MMP9TDP1L3MBTL1MME
SCHEMBL14947768 0.79 PPARG (0.41)
SCHEMBL16261558 0.78 CTNNB1 (0.54) CTNNB1MMP9TDP1L3MBTL1TACR1
SCHEMBL16450886 0.78 CTNNB1 (0.54) CTNNB1MMP9TDP1L3MBTL1TACR1
SCHEMBL14950912 0.78 ALDH1A1 (0.45)
SCHEMBL15686536 0.78 CTNNB1 (0.54) CTNNB1MMP9TDP1L3MBTL1TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017136708-A1 SYNTHESIS AND COMPOSITION OF RAPAFUCIN LIBRARIES THE JOHNS HOPKINS UNIVERSITY (US) 2017-08-10 WO disclosed