SCHEMBL19230614

SCHEMBL19230614

COC(=O)c1ccc2c(c1)CCC(c1ccc(OC)cc1)O2

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.50
ESR2 Q92731 1/20 0.50
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
GABRA1 P14867 2/20 0.46
GABRB2 P47870 2/20 0.46
MAOB P27338 3/20 0.45
CYP19A1 P11511 2/20 0.45
CYP3A4 P08684 1/20 0.45
CYP1A1 P04798 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP1B1 Q16678 1/20 0.44
SLC8A1 P32418 9/20 0.44
NPC1 O15118 1/20 0.43
MAPT P10636 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19230616 0.89 ESR2 (0.65) ESR1ESR2CA1CA2CYP19A1
SCHEMBL19230991 0.84 SLC8A1 (0.43) CA1CA2GABRA1GABRB2CYP19A1
SCHEMBL31395247 0.84 SLC6A4 (0.49) ESR1ESR2
SCHEMBL19230577 0.83 KDM4E (0.44) CA1CA2GABRA1GABRB2SLC8A1
SCHEMBL19230789 0.83 ESR1 (0.39) ESR1ESR2CA1CA2GABRA1
SCHEMBL19230687 0.82 ESR1 (0.46) ESR1ESR2SLC8A1
SCHEMBL7202314 0.81 ESR1 (0.76) ESR1ESR2GABRA1GABRB2MAOB
SCHEMBL19230824 0.81 NOTUM (0.43) SLC8A1
SCHEMBL11047047 0.79 ESR1 (0.52) ESR1ESR2GABRA1GABRB2MAOB
SCHEMBL11049466 0.79 ESR1 (0.56) ESR1ESR2GABRA1GABRB2MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602811-B FXR receptor agonists 轩竹生物科技有限公司 2021-11-16 CN disclosed
WO-2017133521-A1 FXR RECEPTOR AGONIST 山东轩竹医药科技有限公司 2017-08-10 WO disclosed