SCHEMBL19251327

SCHEMBL19251327

CCCCC(C)(C)c1cnc(N)nc1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 11/20 0.37
CNR1 P21554 8/20 0.37
NUDT1 P36639 1/20 0.35
TLR8 Q9NR97 5/20 0.34
PKM P14618 1/20 0.33
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
TLR7 Q9NYK1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18935497 0.93 CNR2 (0.44) CNR2CNR1
SCHEMBL18935596 0.88 NUDT1 (0.37) CNR2NUDT1
SCHEMBL21789887 0.82 CNR2 (0.40) CNR2CNR1ESR1ESR2
SCHEMBL19251008 0.81 NUDT1 (0.33) NUDT1TLR8PKMESR1ESR2
SCHEMBL20017163 0.81 NUDT1 (0.33) CNR2CNR1NUDT1TLR8PKM
SCHEMBL24486521 0.81 CNR2 (0.36) CNR2CNR1TLR8ESR1ESR2
SCHEMBL19251098 0.80 CNR2 (0.35) CNR2CNR1NUDT1TLR8TLR7
SCHEMBL20243849 0.80 CNR2 (0.35) CNR2CNR1NUDT1TLR8TLR7
SCHEMBL19251241 0.79 NPC1 (0.41) NUDT1
SCHEMBL23957925 0.79 NUDT1 (0.34) CNR2CNR1NUDT1TLR8PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9732083-B2 Tricyclic gyrase inhibitors MERCK SHARP & DOHME CORP. (US) 2017-08-15 US disclosed