SCHEMBL19252597

SCHEMBL19252597

CCC(C)(C)c1ccc2c(c1)C(=O)NC2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.50
NPC1 O15118 1/20 0.50
LMNA P02545 1/20 0.50
CASP3 P42574 1/20 0.50
RAB9A P51151 1/20 0.50
ATM Q13315 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
SENP8 Q96LD8 1/20 0.50
SENP7 Q9BQF6 1/20 0.50
SENP6 Q9GZR1 1/20 0.50
CLK4 Q9HAZ1 3/20 0.46
DYRK1B Q9Y463 2/20 0.46
NTRK2 Q16620 2/20 0.46
TYRO3 Q06418 1/20 0.46
FYN P06241 1/20 0.46
NTRK1 P04629 2/20 0.45
FLT3 P36888 2/20 0.45
GSK3B P49841 2/20 0.45
JAK2 O60674 1/20 0.45
MET P08581 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12727793 0.88 NPC1 (0.50) MAPK1NPC1LMNACASP3RAB9A
SCHEMBL19251116 0.85 PARP10 (0.64) MAPK1NPC1LMNACASP3RAB9A
SCHEMBL12220207 0.83 CLK4 (0.51) NPC1CASP3RAB9ASENP8SENP7
SCHEMBL27086074 0.81 PARP1 (0.50) CLK4DYRK1BNTRK2TYRO3FYN
SCHEMBL29871724 0.81 CLK4 (0.49) CLK4DYRK1BNTRK2TYRO3FYN
SCHEMBL10061001 0.79 TDP2 (0.56) MAPK1NPC1LMNACASP3RAB9A
SCHEMBL22886507 0.78 CLK4 (0.39) MAPK1NPC1LMNACASP3RAB9A
SCHEMBL10060999 0.77 NPC1 (0.42) MAPK1NPC1LMNACASP3RAB9A
SCHEMBL30681290 0.77 PARP10 (0.71) CLK4DYRK1BNTRK2TYRO3FYN
SCHEMBL10269253 0.77 MAPK1 (0.46) MAPK1NPC1LMNACASP3RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9732083-B2 Tricyclic gyrase inhibitors MERCK SHARP & DOHME CORP. (US) 2017-08-15 US disclosed