SCHEMBL19258542

SCHEMBL19258542

CC(C)c1ccc(C=N)nc1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TYR P14679 1/20 0.34
NPC1 O15118 2/20 0.33
LMNA P02545 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
KMT2A Q03164 1/20 0.33
RELA Q04206 1/20 0.33
CHRNA7 P36544 1/20 0.31
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL934018 0.79 TYR (0.48) TYRNPC1LMNARAB9ASMN1; SMN2
SCHEMBL13602061 0.70 CCR1 (0.46) TYRNPC1LMNARAB9ASMN1; SMN2
SCHEMBL20621292 0.69 CHRNA7 (0.33) TYRLMNAALDH1A1CHRNA7
SCHEMBL2741630 0.69 ESR1 (0.38) TYRNPC1LMNARAB9ASMN1; SMN2
SCHEMBL179333 0.69 LMNA (0.50) TYRNPC1LMNARAB9ASMN1; SMN2
SCHEMBL15614472 0.68 KRAS (0.34) TYRNPC1LMNARAB9ASMN1; SMN2
SCHEMBL14116462 0.68 ESR1 (0.35) TYRNPC1LMNARAB9ASMN1; SMN2
SCHEMBL25393082 0.68 DHFR (0.37) NPC1LMNARAB9ASMN1; SMN2KDM4E
SCHEMBL25393080 0.68 DHFR (0.37) NPC1LMNARAB9ASMN1; SMN2KDM4E
SCHEMBL15360260 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017133657-A1 PYRIDINE AND PYRIMIDINE DERIVATIVES AND THEIR USE IN TREATMENT, AMELIORATION OR PREVENTION OF INFLUENZA SAVIRA PHARMACEUTICALS GMBH (AT) 2017-08-10 WO disclosed