SCHEMBL19258550

SCHEMBL19258550

C/N=C\c1ncc(C)cc1C

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.43
NOS1 P29475 1/20 0.43
NOS2 P35228 1/20 0.43
CCR1 P32246 1/20 0.34
CCR5 P51681 1/20 0.34
CCR8 P51685 1/20 0.34
CYP2A6 P11509 1/20 0.32
CYP1A2 P05177 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2083611 0.82 NOS3 (0.42) NOS3NOS1NOS2CCR1CCR5
SCHEMBL2083609 0.82 NOS3 (0.42) NOS3NOS1NOS2CCR1CCR5
SCHEMBL20852900 0.79 RRM2 (0.32) NOS3NOS1NOS2CCR1CCR5
SCHEMBL661675 0.76 NOS3 (0.48) NOS3NOS1NOS2CCR1CCR5
SCHEMBL1206724 0.74 NOS3 (0.46) NOS3NOS1NOS2CCR1CCR5
SCHEMBL7245034 0.74 NOS3 (0.46) NOS3NOS1NOS2CCR1CCR5
SCHEMBL7235622 0.72 NOS2 (0.45) NOS3NOS1NOS2CCR1CCR5
SCHEMBL7235627 0.72 NOS2 (0.45) NOS3NOS1NOS2CCR1CCR5
SCHEMBL24861541 0.71
SCHEMBL19937127 0.69 NOS3 (0.42) NOS3NOS1NOS2CCR1CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017133657-A1 PYRIDINE AND PYRIMIDINE DERIVATIVES AND THEIR USE IN TREATMENT, AMELIORATION OR PREVENTION OF INFLUENZA SAVIRA PHARMACEUTICALS GMBH (AT) 2017-08-10 WO disclosed