SCHEMBL19280398

SCHEMBL19280398

CC1CN(C(=O)O)CC(C)N1c1cccc(Br)c1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.45
ADAMTS5 Q9UNA0 1/20 0.40
OPRM1 P35372 1/20 0.40
ALKBH5 Q6P6C2 1/20 0.40
ALDH1A1 P00352 2/20 0.40
TP53 P04637 1/20 0.40
SLC6A9 P48067 2/20 0.39
AR P10275 1/20 0.39
KMT5A Q9NQR1 1/20 0.38
MGLL Q99685 3/20 0.38
HPGD P15428 1/20 0.38
POLB P06746 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
ATM Q13315 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
L3MBTL3 Q96JM7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19690265 0.88 ALOX5 (0.45) ALOX5ADAMTS5ALDH1A1TP53AR
SCHEMBL19690264 0.88 ALOX5 (0.45) ALOX5ADAMTS5ALDH1A1TP53AR
SCHEMBL18043595 0.84 NOTUM (0.52) ALOX5ALDH1A1TP53ARPOLB
SCHEMBL18043606 0.82 AR (0.47) ALOX5OPRM1ALDH1A1ARHPGD
SCHEMBL19385695 0.82 AR (0.47) ALOX5OPRM1ALDH1A1ARHPGD
SCHEMBL23777680 0.82 ADAMTS5 (0.54) ADAMTS5ALDH1A1TP53MGLLHPGD
SCHEMBL11963050 0.82 ADAMTS5 (0.54) ADAMTS5ALDH1A1TP53MGLLHPGD
SCHEMBL23777797 0.82 ADAMTS5 (0.54) ADAMTS5ALDH1A1TP53MGLLHPGD
SCHEMBL19690137 0.81 USP30 (0.50) ALOX5
SCHEMBL19690138 0.81 USP30 (0.50) ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3209664-A1 BICYCLIC HETEROARYL AMINE COMPOUNDS AS PI3K INHIBITORS Bristol-Myers Squibb Company (US) 2017-08-30 EP disclosed