SCHEMBL19288091

SCHEMBL19288091

C=C(N)CCNC(=O)c1cc(NC(=O)c2cc(NC(=O)CNC(=N)N)cn2C)cn1C

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 2/20 0.62
HRAS P01112 14/20 0.60
ESR1 P03372 13/20 0.60
ESR2 Q92731 13/20 0.60
KDM4E B2RXH2 1/20 0.59
POLB P06746 1/20 0.59
MAPT P10636 1/20 0.59
HIF1A Q16665 1/20 0.59
HDAC1 Q13547 2/20 0.40
HDAC2 Q92769 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
ERBB2 P04626 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14267762 0.91 TOP1 (0.74) TOP1HRASESR1ESR2KDM4E
Netropsin SCHEMBL197747 0.91 TOP1 (0.74) TOP1HRASESR1ESR2KDM4E
Netropsin SCHEMBL4953090 0.90 TOP1 (0.72) TOP1HRASESR1ESR2KDM4E
Netropsin SCHEMBL10408939 0.90 TOP1 (0.72) TOP1HRASESR1ESR2KDM4E
Netropsin SCHEMBL951644 0.89 TOP1 (0.71) TOP1HRASESR1ESR2KDM4E
SCHEMBL12348338 0.89 TOP1 (0.70) TOP1HRASESR1ESR2KDM4E
SCHEMBL12348157 0.87 TOP1 (0.65) TOP1HRASESR1ESR2KDM4E
Netropsin SCHEMBL4284668 0.81 TOP1 (0.60) TOP1HRASESR1ESR2KDM4E
SCHEMBL12628472 0.80 TOP1 (0.48) TOP1HRASESR1ESR2KDM4E
Netropsin SCHEMBL4955084 0.78 TOP1 (0.56) TOP1HRASESR1ESR2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9745337-B2 Complex compounds of germanium, methods for producing same, and drugs OBSCHESNO S OGRANICHENNOI OTVETSTVENNOSTYU “WDS FARMA” (RU) 2017-08-29 US disclosed