SCHEMBL19289751

SCHEMBL19289751

Cc1cccc(C(C)C)c1C[C@H](C)N

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.48
GABRG2 P18507 2/20 0.48
GABRB3 P28472 2/20 0.48
TAAR1 Q96RJ0 4/20 0.45
MAOA P21397 3/20 0.45
SLC6A2 P23975 3/20 0.45
SLC6A4 P31645 2/20 0.45
SLC6A3 Q01959 1/20 0.45
SIGMAR1 Q99720 1/20 0.45
CYP2A6 P11509 1/20 0.45
ADORA2A P29274 1/20 0.45
ADORA1 P30542 1/20 0.45
SCN4A P35499 3/20 0.43
LMNA P02545 3/20 0.43
HTR2B P41595 3/20 0.43
HTR2A P28223 2/20 0.43
SCN1A P35498 2/20 0.43
SCN5A Q14524 2/20 0.43
SCN9A Q15858 2/20 0.43
CYP1A2 P05177 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13692287 0.86 SLC6A2 (0.54) TAAR1MAOASLC6A2SLC6A4SLC6A3
SCHEMBL16273856 0.84 GABRA1 (0.44) GABRA1GABRG2GABRB3TAAR1MAOA
Hydrochloric Acid SCHEMBL29444026 0.84 TAAR1 (0.52) TAAR1MAOASLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL28478337 0.84 TAAR1 (0.52) TAAR1MAOASLC6A2SLC6A4SLC6A3
SCHEMBL3865790 0.80 GABRA1 (0.52) GABRA1GABRG2GABRB3TAAR1MAOA
SCHEMBL9734713 0.78 GABRA1 (0.54) GABRA1GABRG2GABRB3TAAR1MAOA
SCHEMBL19289757 0.77 GABRA1 (0.48) GABRA1GABRG2GABRB3TAAR1MAOA
SCHEMBL6215211 0.76 GABRA1 (0.52) GABRA1GABRG2GABRB3TAAR1MAOA
SCHEMBL6213612 0.76 GABRA1 (0.76) GABRA1GABRG2GABRB3TAAR1SLC6A2
SCHEMBL5823486 0.76 GABRA1 (0.52) GABRA1GABRG2GABRB3TAAR1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3004061-B1 3,4-DIHYDROISOQUINOLIN-2(1H)-YL COMPOUNDS LILLY CO ELI (US) 2017-08-30 EP disclosed