SCHEMBL19308657

SCHEMBL19308657

O=C(O)N1CCC(n2ccnc2-c2ccc(Cl)cc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
F10 P00742 3/20 0.43
ABCC9 O60706 2/20 0.39
MGLL Q99685 4/20 0.38
MAPT P10636 1/20 0.38
HRH3 Q9Y5N1 1/20 0.37
SLC6A7 Q99884 1/20 0.36
HTR2B P41595 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
AKR1C3 P42330 1/20 0.35
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
SPR P35270 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3564565 0.88 ESR1 (0.43) F10ABCC9HTR2B
SCHEMBL16827710 0.81 PDK2 (0.52)
SCHEMBL16845847 0.79 CNR1 (0.39) F10ABCC9CNR1CNR2
SCHEMBL3560855 0.73 GPR119 (0.53)
SCHEMBL28226097 0.71 ESR1 (0.41) ABCC9MAPTKMT2A
SCHEMBL16828064 0.71 PDK2 (0.53)
SCHEMBL2464307 0.71 DYRK1A (0.43)
SCHEMBL27277040 0.70 PDE4A (0.44) ABCC9MEN1KMT2A
SCHEMBL4991364 0.68 HRH3 (0.47) F10MAPTHRH3
SCHEMBL27761911 0.67 LMNA (0.43) ABCC9MAPTCNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9751861-B2 N1-(3,3,3-trifluoro-2-hydroxo-2-methylpropionyl)-piperidine derivatives as inhibitors of pyruvate dehydrogenase kinase MERCK PATENT GMBH (DE) 2017-09-05 US disclosed