SCHEMBL19320897

SCHEMBL19320897

COCc1ccccc1-n1nc2c(c1C(=O)O)CC(C(F)(F)F)CC2

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CACNA1G O43497 1/20 0.37
CACNA1H O95180 1/20 0.37
CACNA1I Q9P0X4 1/20 0.37
RIPK1 Q13546 4/20 0.35
SIGMAR1 Q99720 5/20 0.34
ENPP2 Q13822 1/20 0.34
TMEM97 Q5BJF2 4/20 0.33
POLQ O75417 3/20 0.33
ADRA1A P35348 1/20 0.33
NTRK1 P04629 2/20 0.31
TP53 P04637 1/20 0.31
PRMT5 O14744 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19320901 0.91 TP53 (0.39) RIPK1SIGMAR1TMEM97ADRA1ATP53
SCHEMBL19325551 0.90 CACNA1G (0.35) CACNA1GCACNA1HCACNA1IRIPK1SIGMAR1
SCHEMBL19320900 0.86 HCAR2 (0.39) RIPK1SIGMAR1TMEM97ADRA1APRMT5
SCHEMBL19320898 0.83 RIPK1 (0.42) CACNA1GCACNA1HCACNA1IRIPK1SIGMAR1
SCHEMBL19325964 0.83 TP53 (0.38) RIPK1SIGMAR1TMEM97TP53
SCHEMBL19325960 0.77 HCAR2 (0.39) RIPK1SIGMAR1TMEM97ADRA1A
SCHEMBL19320896 0.76 CACNA1G (0.42) CACNA1GCACNA1HCACNA1I
SCHEMBL19320827 0.74 CYP3A4 (0.32) CACNA1GCACNA1HCACNA1I
SCHEMBL19325528 0.74 RIPK1 (0.41) CACNA1GCACNA1HCACNA1IRIPK1SIGMAR1
SCHEMBL18366104 0.72 POLB (0.54) CACNA1GCACNA1HCACNA1IRIPK1POLQ

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170253607-A1 LONG-ACTING HIV PROTEASE INHIBITOR SHIONOGI & CO., LTD. (JP) 2017-09-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170253607-A1 LONG-ACTING HIV PROTEASE INHIBITOR CPN1, HAT1, PRSS1 CACNA1G 3034/4885CACNA1H 2888/4885CACNA1I 2662/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.