SCHEMBL19328

SCHEMBL19328

CCOC(=O)c1c(C)n[nH]c1C(F)F

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 1/20 0.65
KDM4E B2RXH2 6/20 0.43
MAPT P10636 3/20 0.43
POLB P06746 2/20 0.43
KMT2A Q03164 2/20 0.43
LMNA P02545 3/20 0.39
PKM P14618 1/20 0.39
HPGD P15428 4/20 0.39
ALDH1A1 P00352 7/20 0.39
SMN1; SMN2 Q16637 5/20 0.39
GAA P10253 3/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
NPSR1 Q6W5P4 2/20 0.38
RAB9A P51151 2/20 0.38
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15165757 0.86 PDE4D (0.50) PDE4DKDM4EMAPTPOLBKMT2A
SCHEMBL14812013 0.85 PDE4D (0.67) PDE4DKDM4EMAPTPOLBKMT2A
SCHEMBL2084738 0.84 SMN1; SMN2 (0.50) PDE4DKDM4EMAPTPOLBKMT2A
SCHEMBL20583553 0.84 PDE4D (0.49) PDE4DKDM4EMAPTPOLBKMT2A
SCHEMBL28350936 0.84 PDE4D (0.65) PDE4DKDM4EMAPTPOLBKMT2A
SCHEMBL28112151 0.83 PDE4D (0.42) PDE4DKDM4EMAPTPOLBKMT2A
SCHEMBL4650693 0.82 KDM4E (0.52) PDE4DKDM4EMAPTPOLBKMT2A
SCHEMBL20075372 0.79 PDE4D (0.39) PDE4DKDM4ELMNAALDH1A1NPSR1
SCHEMBL353564 0.79 PDE4D (1.00) PDE4DKDM4EMAPTPOLBKMT2A
SCHEMBL22637869 0.78 PDE4D (0.38) PDE4DKDM4EKMT2ALMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106467492-B preparation method of polyfluoromethyl pyrazole compound, intermediate and preparation method 联化科技(盐城)有限公司 2019-12-17 CN disclosed
WO-2014033164-A1 PROCEDURE FOR THE DECARBOXYLATION OF 3,5-BIS(HALOALKYL)-PYRAZOLE-4-CARBOXYLIC ACID DERIVATIVES BAYER CROPSCIENCE AG (DE) 2014-03-06 WO disclosed
WO-2012025469-A1 IMPROVED PROCESS FOR THE PREPARATION OF ESTERS OF 1-H-PYRAZOLE-4-CARBOXYLIC ACIDS SOLVAY SA (BE) 2012-03-01 WO disclosed