SCHEMBL1932974

SCHEMBL1932974

COc1ccc(-c2cc3nc(CC=O)cnc3n2COCC[Si](C)(C)C)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 3/20 0.34
TDP1 Q9NUW8 1/20 0.34
DGAT1 O75907 3/20 0.33
CYP1A2 P05177 7/20 0.33
CYP3A4 P08684 5/20 0.33
CYP2C9 P11712 3/20 0.33
CYP2D6 P10635 2/20 0.33
CYP2C19 P33261 2/20 0.33
ALDH1A1 P00352 9/20 0.33
USP2 O75604 7/20 0.33
CASP1 P29466 7/20 0.33
CASP7 P55210 7/20 0.33
HSD17B10 Q99714 7/20 0.33
HIF1A Q16665 4/20 0.33
TSHR P16473 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
MAPT P10636 2/20 0.32
HPGD P15428 2/20 0.32
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2314920 0.83 DGAT1 (0.38) ALOX15TDP1DGAT1CYP1A2CYP3A4
SCHEMBL1932973 0.82 DGAT1 (0.39) ALOX15TDP1DGAT1ALDH1A1HSD17B10
SCHEMBL2317159 0.79 TDP1 (0.39) ALOX15TDP1DGAT1ALDH1A1USP2
SCHEMBL4065268 0.74 TDP1 (0.44) ALOX15TDP1DGAT1ALDH1A1USP2
SCHEMBL1536819 0.73 LCK (0.38) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL2320195 0.72 ALOX15 (0.37) ALOX15TDP1DGAT1ALDH1A1USP2
SCHEMBL1536984 0.72 LCK (0.39) CYP1A2CYP3A4CYP2C9USP2CASP1
SCHEMBL1536781 0.72 LCK (0.39) CYP1A2CYP3A4CYP2C9CYP2C19USP2
SCHEMBL2315378 0.71 TDP1 (0.36) ALOX15TDP1DGAT1ALDH1A1USP2
SCHEMBL2317903 0.71 LCK (0.39) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2506713-A1 NOVEL TRICYCLIC COMPOUNDS Abbott Laboratories (US) 2012-10-10 EP disclosed
WO-2011068899-A1 NOVEL TRICYCLIC COMPOUNDS ABBOTT LABORATORIES (US) 2011-06-09 WO disclosed