SCHEMBL19334390

SCHEMBL19334390

Cc1ccccc1NCC(=O)N/N=C\c1cc([N+](=O)O)cc(Br)c1O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 7/20 0.58
KMT2A Q03164 7/20 0.58
MAPT P10636 9/20 0.53
ALDH1A1 P00352 5/20 0.53
SMN1; SMN2 Q16637 3/20 0.53
GAA P10253 1/20 0.53
HTT P42858 5/20 0.52
TDP1 Q9NUW8 3/20 0.52
GRK2 P25098 1/20 0.50
CFTR P13569 1/20 0.50
ERCC1 P07992 1/20 0.50
ERCC4 Q92889 1/20 0.50
LMNA P02545 7/20 0.49
LIG1 P18858 2/20 0.49
LIG3 P49916 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
POLB P06746 1/20 0.49
KDM4E B2RXH2 3/20 0.48
HPGD P15428 2/20 0.48
MAPK1 P28482 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13401793 0.91 MEN1 (0.67) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL12648536 0.85 CFTR (0.67) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL14082236 0.82 MAPT (0.58) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL13401808 0.77 MAPT (0.57) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL14959214 0.77 MAPT (0.59) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL19334398 0.75 MAPT (0.58) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL19334394 0.74 ALDH1A1 (0.59) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL16211083 0.73 KDM4E (0.67) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL16211082 0.73 KDM4E (0.67) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL19334492 0.73 LIG1 (0.62) MEN1KMT2AMAPTALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9757375-B2 Compounds that inhibit human DNA ligases and methods of treating cancer UNIVERSITY OF MARYLAND, BALTIMORE (US) 2017-09-12 US disclosed